SCHEMBL8964634

SCHEMBL8964634

COc1ccc(COC=CCc2ccc(OCc3ccc(OC)cc3)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
APP P05067 7/20 0.56
MAOB P27338 1/20 0.54
SMN1; SMN2 Q16637 2/20 0.50
NPC1 O15118 2/20 0.50
RAB9A P51151 2/20 0.50
POLB P06746 1/20 0.50
IDO1 P14902 2/20 0.49
AGXT P21549 2/20 0.49
FFAR1 O14842 1/20 0.48
ALDH1A1 P00352 2/20 0.47
TP53 P04637 1/20 0.47
CYP3A4 P08684 1/20 0.47
ALOX15 P16050 1/20 0.47
TSHR P16473 1/20 0.47
ALOX12 P18054 1/20 0.47
MAPT P10636 1/20 0.47
HTT P42858 1/20 0.47
TDP1 Q9NUW8 1/20 0.46
PLA2G4B P0C869 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8964654 0.86 NPC1 (0.56) APPMAOBNPC1RAB9ATDP1
SCHEMBL20000873 0.80 APP (0.80) APPMAOBSMN1; SMN2NPC1RAB9A
SCHEMBL933579 0.80 APP (0.62) APPMAOBSMN1; SMN2NPC1RAB9A
SCHEMBL9797652 0.78 SMN1; SMN2 (0.79) APPMAOBSMN1; SMN2NPC1RAB9A
SCHEMBL5598799 0.77 ALDH1A1 (0.59) MAOBSMN1; SMN2IDO1AGXTALDH1A1
SCHEMBL7921584 0.77 ALDH1A1 (0.59) MAOBSMN1; SMN2IDO1AGXTALDH1A1
SCHEMBL6550928 0.77 IDO1 (0.52) APPMAOBSMN1; SMN2NPC1RAB9A
SCHEMBL11437812 0.76 ALDH1A1 (0.68) MAOBSMN1; SMN2IDO1AGXTALDH1A1
SCHEMBL8964668 0.76 IDO1 (0.44) APPMAOBSMN1; SMN2NPC1RAB9A
SCHEMBL8965482 0.76 IDO1 (0.44) APPMAOBSMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed