SCHEMBL8964654

SCHEMBL8964654

COc1ccc(COC=CCc2cccc(OCc3ccc(OC)cc3)c2)cc1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.56
RAB9A P51151 1/20 0.56
TDP1 Q9NUW8 1/20 0.56
MAOB P27338 10/20 0.54
BCHE P06276 2/20 0.52
APP P05067 1/20 0.50
TLR4 O00206 1/20 0.48
TLR2 O60603 1/20 0.48
SMPD1 P17405 1/20 0.48
ABCB1 P08183 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8964634 0.86 APP (0.56) NPC1RAB9ATDP1MAOBAPP
SCHEMBL28567450 0.82 ALDH1A1 (0.60) NPC1RAB9ATDP1MAOBBCHE
SCHEMBL13462938 0.78 MAOB (0.65) NPC1RAB9ATDP1MAOBBCHE
SCHEMBL10820376 0.78 MAOB (0.67) NPC1RAB9ATDP1MAOBBCHE
SCHEMBL7813380 0.77 MAOB (0.63) NPC1RAB9ATDP1MAOBBCHE
SCHEMBL8965482 0.75 IDO1 (0.44) NPC1RAB9ATDP1MAOBBCHE
SCHEMBL8964668 0.75 IDO1 (0.44) NPC1RAB9ATDP1MAOBAPP
SCHEMBL28084246 0.75 IDO1 (0.56) MAOB
SCHEMBL24041859 0.74 CYP4F2 (0.74) NPC1RAB9ATDP1MAOBBCHE
SCHEMBL10819608 0.74 NPC1 (0.61) NPC1RAB9ATDP1MAOBBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed