SCHEMBL8964647

SCHEMBL8964647

C=CCc1cc(OCc2ccc(OC)cc2)cc(OCc2ccc(OC)cc2)c1

nearest known ligand 0.66

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.66
SMN1; SMN2 Q16637 2/20 0.66
TP53 P04637 1/20 0.66
CYP3A4 P08684 1/20 0.66
ALOX15 P16050 1/20 0.66
TSHR P16473 1/20 0.66
ALOX12 P18054 1/20 0.66
APP P05067 6/20 0.51
MAOB P27338 5/20 0.50
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
TDP1 Q9NUW8 1/20 0.49
FFAR4 Q5NUL3 1/20 0.48
PPARG P37231 2/20 0.47
PPARD Q03181 2/20 0.47
PPARA Q07869 2/20 0.47
FFAR1 O14842 1/20 0.47
POLB P06746 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9797652 0.88 SMN1; SMN2 (0.79) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
SCHEMBL28567450 0.86 ALDH1A1 (0.60) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
SCHEMBL8965477 0.82 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
SCHEMBL8964657 0.82 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
SCHEMBL8964626 0.81 ALDH1A1 (0.62) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
SCHEMBL1514243 0.80 ALDH1A1 (0.63) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
Estragole SCHEMBL28095175 0.80 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
Estragole SCHEMBL57204 0.80 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
Estragole SCHEMBL900647 0.80 ALDH1A1 (1.00) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15
SCHEMBL8964769 0.79 ALDH1A1 (0.58) ALDH1A1SMN1; SMN2TP53CYP3A4ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed