SCHEMBL8965460

SCHEMBL8965460

C=CCc1cc(C)c(OC)c(C)c1

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FFAR4 Q5NUL3 1/20 0.49
ALDH1A1 P00352 5/20 0.48
PPARG P37231 1/20 0.48
PPARD Q03181 1/20 0.48
PPARA Q07869 1/20 0.48
CYP3A4 P08684 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
ALOX15 P16050 2/20 0.48
TP53 P04637 1/20 0.48
TSHR P16473 1/20 0.48
ALOX12 P18054 1/20 0.48
PTGS1 P23219 2/20 0.44
ALOX5 P09917 2/20 0.44
AR P10275 1/20 0.44
TRPM8 Q7Z2W7 1/20 0.44
TNKS O95271 1/20 0.44
TNKS2 Q9H2K2 1/20 0.44
GABRA1 P14867 2/20 0.40
GABRB2 P47870 2/20 0.40
MAPT P10636 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16313803 0.89 FFAR4 (0.44) FFAR4ALDH1A1PPARGPPARDPPARA
SCHEMBL3141953 0.89 ALDH1A1 (0.56) FFAR4ALDH1A1PPARGPPARDPPARA
SCHEMBL22689193 0.87 TNKS (0.53) FFAR4ALDH1A1PPARGPPARDPPARA
SCHEMBL23230324 0.82 FFAR4 (0.41) FFAR4ALDH1A1PPARGPPARDPPARA
SCHEMBL17438120 0.81 FFAR4 (0.38) FFAR4ALDH1A1PPARGPPARDPPARA
SCHEMBL770139 0.81 ALDH1A1 (0.50) ALDH1A1PPARGPPARDPPARACYP3A4
SCHEMBL4784297 0.81 ALDH1A1 (0.42) FFAR4ALDH1A1DHFR
SCHEMBL5082696 0.80 FFAR4 (0.40) FFAR4ALDH1A1PPARGPPARDPPARA
SCHEMBL68542 0.79 ALDH1A1 (0.63) ALDH1A1PPARGPPARDPPARACYP3A4
SCHEMBL9155768 0.79 FFAR4 (0.39) FFAR4ALDH1A1PPARGPPARDPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0410379-B1 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMA (US) 1996-01-31 EP disclosed
US-5068465-A Hypotensive agents or enzyme inhibitors for treatment of hypertension MERRELL DOW PHARMACEUTICALS INC. (US) 1991-11-26 US disclosed
EP-0410379-A2 Pharmaceutically active 3-aryl and 3-heteroaryl-2-fluoro-1-olefins MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-30 EP disclosed
US-4981868-A ENZYME INHIBITORS, HYPOTENSIVES MERRELL DOW PHARMACEUTICAL (US) 1991-01-01 US disclosed