SCHEMBL8965862

SCHEMBL8965862

COc1cc(CO)c2ccccc2c1

nearest known ligand 0.51

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 1/20 0.50
CDC25B P30305 4/20 0.49
MEN1 O00255 1/20 0.49
KMT2A Q03164 1/20 0.49
CYP1A2 P05177 1/20 0.48
CYP2A6 P11509 1/20 0.48
TDP1 Q9NUW8 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
MTNR1A P48039 1/20 0.44
MTNR1B P49286 1/20 0.44
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
NQO1 P15559 1/20 0.42
NQO2 P16083 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13490711 0.85 CDC25B (0.49) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL21822099 0.84 L3MBTL1 (0.49) CYP1A2L3MBTL1MTNR1BNQO1NQO2
SCHEMBL15345649 0.84 MEN1 (0.48) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL5252235 0.84 MEN1 (0.48) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL4699483 0.84 MEN1 (0.48) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL4702310 0.84 MEN1 (0.48) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL30747862 0.83 GRM5 (0.37) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL29151462 0.83 GRM5 (0.37) AKR1B1CDC25BMEN1KMT2ACYP1A2
SCHEMBL6856603 0.82 MTNR1A (0.59) CYP1A2CYP2A6TDP1L3MBTL1MTNR1A
SCHEMBL20562784 0.81 TAAR1 (0.51) AKR1B1MEN1KMT2ACYP1A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed
US-5371219-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1994-12-06 US disclosed
EP-0305093-B1 Imidazo(1,2-b)pyridazine derivatives WELLCOME FOUND (GB) 1994-04-06 EP disclosed
US-5091531-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1992-02-25 US disclosed
EP-0305093-A1 Imidazo(1,2-b)pyridazine derivatives THE WELLCOME FOUNDATION LIMITED (GB) 1989-03-01 EP disclosed