SCHEMBL8965978

SCHEMBL8965978

COC(=O)Nc1cn2nc(OCc3cc(OC)c(OCOC(C)OC)c(OC)c3)ccc2n1

nearest known ligand 0.78

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 4/20 0.40
KDR P35968 10/20 0.36
RIPK1 Q13546 4/20 0.36
CSNK1D P48730 1/20 0.35
MET P08581 1/20 0.35
PIK3CD O00329 1/20 0.34
PIK3CG P48736 1/20 0.34
AURKA O14965 1/20 0.34
PDGFRB P09619 1/20 0.34
KIT P10721 1/20 0.34
FLT1 P17948 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9373529 0.93 PIK3CA (0.41) PIK3CAKDRRIPK1CSNK1DMET
SCHEMBL8965590 0.88 PIK3CA (0.45) PIK3CAKDRRIPK1CSNK1DMET
SCHEMBL8965977 0.87 PIK3CA (0.44) PIK3CAKDRRIPK1CSNK1DMET
SCHEMBL8965975 0.85 PIK3CA (0.45) PIK3CAKDRRIPK1METPIK3CD
SCHEMBL8965973 0.84 PIK3CA (0.39) PIK3CAKDRRIPK1CSNK1DMET
SCHEMBL8965640 0.81 KDR (0.44) PIK3CAKDRCSNK1DMETPIK3CD
SCHEMBL8965644 0.81 PIK3CA (0.42) PIK3CAKDRRIPK1CSNK1DMET
SCHEMBL8965523 0.80 PIK3CA (0.47) PIK3CAKDRRIPK1CSNK1DMET
SCHEMBL8965909 0.80 PIK3CA (0.42) PIK3CAKDRRIPK1PIK3CDPIK3CG
SCHEMBL9369315 0.80 PIK3CA (0.46) PIK3CAKDRRIPK1METPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5538970-A Treatment of cancer with imidazo-1,2-pyridazin compounds GLAXO WELLCOME INC. (US) 1996-07-23 US disclosed
US-5447956-A Anticarcinogenic agents BURROUGHS WELLCOME CO. (US) 1995-09-05 US disclosed