SCHEMBL8966528

SCHEMBL8966528

COc1c(C(=O)NCCNC2CCCCC2)cc(N)c2ccccc12

nearest known ligand 0.50

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 18/20 0.50
DRD3 P35462 1/20 0.48
CNR1 P21554 1/20 0.46
CNR2 P34972 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967329 1.00 SIGMAR1 (0.50) SIGMAR1DRD3CNR1CNR2
Hydrochloric Acid SCHEMBL8967140 0.99 SIGMAR1 (0.49) SIGMAR1DRD3CNR1CNR2
Hydrochloric Acid SCHEMBL9223939 0.87 SIGMAR1 (0.52) SIGMAR1DRD3
SCHEMBL8967226 0.87 SIGMAR1 (0.66) SIGMAR1DRD3
SCHEMBL8967338 0.87 DRD3 (0.59) SIGMAR1DRD3
Hydrochloric Acid SCHEMBL9229456 0.87 SIGMAR1 (0.52) SIGMAR1DRD3
Hydrochloric Acid SCHEMBL8966597 0.86 DRD3 (0.58) SIGMAR1DRD3
SCHEMBL8967463 0.85 SIGMAR1 (0.48) SIGMAR1DRD3
SCHEMBL8967296 0.84 DRD3 (0.51) SIGMAR1DRD3
Hydrochloric Acid SCHEMBL8967334 0.83 DRD3 (0.51) SIGMAR1DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585116-B1 1-Alkoxy-naphthalene-2-carboxamide derivatives with high affinity for the serotonin 5-HT1A receptor LILLY INDUSTRIES LTD (GB) 1996-02-28 EP disclosed
US-5389684-A Treats disorder of central nervous system LILLY INDUSTRIES LIMITED (GB) 1995-02-14 US disclosed