SCHEMBL8966737

SCHEMBL8966737

COc1ccc(C(=O)NCCCSc2ccncc2)cc1

nearest known ligand 0.65

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 5/20 0.65
ALDH1A1 P00352 5/20 0.65
RAB9A P51151 4/20 0.65
SMN1; SMN2 Q16637 3/20 0.65
NFKB1 P19838 1/20 0.65
NFKB2 Q00653 1/20 0.65
RELA Q04206 1/20 0.65
HPGD P15428 1/20 0.57
TP53 P04637 1/20 0.56
KMT2A Q03164 3/20 0.55
TSHR P16473 2/20 0.55
MAPT P10636 1/20 0.55
L3MBTL1 Q9Y468 1/20 0.54
MEN1 O00255 1/20 0.53
MTNR1A P48039 1/20 0.51
MTNR1B P49286 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8967166 0.89 NPC1 (0.52) NPC1ALDH1A1RAB9ASMN1; SMN2NFKB1
Hydrochloric Acid SCHEMBL8967090 0.87 SMN1; SMN2 (0.63) NPC1ALDH1A1RAB9ASMN1; SMN2HPGD
SCHEMBL8967975 0.87 NAAA (0.59) NPC1ALDH1A1RAB9ASMN1; SMN2NFKB1
SCHEMBL8966997 0.86 SMN1; SMN2 (0.60) NPC1ALDH1A1RAB9ASMN1; SMN2HPGD
SCHEMBL8967171 0.83 RAB9A (0.66) NPC1ALDH1A1RAB9ASMN1; SMN2NFKB1
Hydrochloric Acid SCHEMBL8966784 0.82 RAB9A (0.57) NPC1ALDH1A1RAB9ASMN1; SMN2NFKB1
Hydrochloric Acid SCHEMBL8966805 0.82 KMT2A (0.52) NPC1RAB9ASMN1; SMN2NFKB1NFKB2
SCHEMBL11755751 0.81 NPC1 (0.77) NPC1ALDH1A1RAB9ASMN1; SMN2NFKB1
Hydrochloric Acid SCHEMBL8966539 0.80 KMT2A (0.59) NPC1ALDH1A1RAB9ASMN1; SMN2NFKB1
Hydrochloric Acid SCHEMBL8967041 0.80 NAAA (0.55) NPC1RAB9ASMN1; SMN2HPGDKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5561147-A ANTIINFLAMMATORY AGENT, ANTIPYRETIC, ANALGESICS, ANTIALLERGENS, IMMUNOSUPPRESSANTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-01 US disclosed
EP-0522606-B1 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1996-04-03 EP disclosed
US-5457106-A Antiinflammatory agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-10-10 US disclosed
US-5389658-A Administering as antipyretic, antiinflammatory, analgesic, antiallergic, or immunosupressive agents TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-02-14 US disclosed
EP-0612729-A2 Pyridine derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1994-08-31 EP disclosed
US-5246948-A Antiinflammatory, antipyretic, analgesic, antiallergic, immunosupressing or immunomodulating activity TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-09-21 US disclosed
EP-0522606-A2 Pyridine derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1993-01-13 EP disclosed