SCHEMBL8966767

SCHEMBL8966767

CCOC(=O)Nc1ccc(NCc2ccccc2)cc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 1/20 0.54
KCNQ2 O43526 1/20 0.54
KCNQ4 P56696 1/20 0.54
KCNQ5 Q9NR82 1/20 0.54
ALDH1A1 P00352 3/20 0.54
L3MBTL1 Q9Y468 2/20 0.52
PKM P14618 2/20 0.52
NPC1 O15118 5/20 0.50
RAB9A P51151 5/20 0.50
CYP2D6 P10635 2/20 0.50
CYP2C9 P11712 2/20 0.50
CYP2C19 P33261 2/20 0.50
TSHR P16473 1/20 0.50
MAPT P10636 8/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
POLB P06746 2/20 0.49
MAPK1 P28482 1/20 0.49
KMT2A Q03164 6/20 0.48
MEN1 O00255 4/20 0.48
HPGD P15428 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2235641 0.89 KCNQ2 (0.70) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL6004934 0.89 MAPT (0.49) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL6004821 0.87 KCNQ3 (0.48) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL17761732 0.87 ALDH1A1 (0.60) ALDH1A1L3MBTL1PKMNPC1RAB9A
SCHEMBL6005078 0.86 KCNQ3 (0.50) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL20134035 0.86 KCNQ3 (0.55) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL8966006 0.86 KCNQ2 (0.58) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL20133977 0.86 KCNQ3 (0.48) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL20133927 0.86 THRB (0.53) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1
SCHEMBL4994653 0.85 ALDH1A1 (0.53) KCNQ3KCNQ2KCNQ4KCNQ5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0554543-B1 1,2,4-Triaminobenzene derivatives and process for their preparation ASTA MEDICA AG (DE) 1996-02-28 EP disclosed
US-5384330-A Pharmaceutically active 1,2,4-triamino-benzene derivatives, processes for their preparation and pharmaceutical compositions containing them ASTA MEDICA AKTIENGESELLSCHAFT (DE) 1995-01-24 US disclosed
EP-0554543-A2 1,2,4-Triaminobenzene derivatives and process for their preparation ASTA Medica Aktiengesellschaft (DE) 1993-08-11 EP disclosed