SCHEMBL896743

SCHEMBL896743

[O-][S@+](Cc1cncc(OCC2CC2)c1)c1nc2cc(F)ccc2[nH]1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.37
CHRNB2 P17787 5/20 0.35
CHRNA4 P43681 3/20 0.35
CHRNA6 Q15825 1/20 0.34
KDM1A O60341 2/20 0.32
CHRNB1 P11230 1/20 0.32
CHRNB4 P30926 1/20 0.32
CHRNA3 P32297 1/20 0.32
CHRNB3 Q05901 1/20 0.32
PDE2A O00408 1/20 0.31
PRMT5 O14744 1/20 0.31
WDR77 Q9BQA1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL896742 1.00 CYP2C9 (0.37) CYP2C9CHRNB2CHRNA4CHRNA6KDM1A
SCHEMBL3381144 0.82 CYP2C9 (0.53) CYP2C9
SCHEMBL9227422 0.82 CYP2C9 (0.52) CYP2C9
SCHEMBL9226291 0.82 CYP2C9 (0.52) CYP2C9
SCHEMBL10034496 0.75 CYP2C9 (0.36) CYP2C9
SCHEMBL6481793 0.71 MAOA (0.34) CYP2C9KDM1APDE2A
SCHEMBL8787879 0.70 CYP2C9 (0.51) CYP2C9
SCHEMBL8435843 0.69 CYP2C9 (0.46) CYP2C9
SCHEMBL6476381 0.69 SLC6A2 (0.35) PDE2A
SCHEMBL10207815 0.68 ATP4A (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8793078-B2 Method for predicting activation energy using atomic fingerprint descriptor or atomic descriptor BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2014-07-29 US disclosed
US-20120084012-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING ATOMIC FINGERPRINT DESCRIPTOR OR ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2012-04-05 US disclosed
US-20110213558-A1 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR BIOINFORMATICS & MOLECULAR DESIGN RESEARCH CENTER (KR) 2011-09-01 US disclosed
EP-2354987-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR Bioinformatics&Molecular Design Research Center (KR) 2011-08-10 EP disclosed
WO-2010056053-A2 METHOD FOR PREDICTING ACTIVATION ENERGY USING AN ATOMIC FINGERPRINT DESCRIPTOR OR AN ATOMIC DESCRIPTOR 사단법인 분자설계연구소 (KR) 2010-05-20 WO disclosed