SCHEMBL8967698

SCHEMBL8967698

OC(CCCN1CC[C@](O)(c2ccccc2)[C@@H](C(O)c2ccccc2)C1)c1ccc(Br)cc1

nearest known ligand 0.63

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.63
TSHR P16473 1/20 0.63
SLC6A3 Q01959 1/20 0.47
KMT2A Q03164 2/20 0.42
LMNA P02545 2/20 0.42
OPRL1 P41146 2/20 0.41
OPRM1 P35372 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
IGF1R P08069 2/20 0.41
MEN1 O00255 1/20 0.41
DRD2 P14416 3/20 0.41
SIGMAR1 Q99720 3/20 0.41
DRD3 P35462 2/20 0.41
SLC18A3 Q16572 1/20 0.40
CCR1 P32246 1/20 0.40
GRIN2B Q13224 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9173912 0.94 ALDH1A1 (0.71) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL8967036 0.90 ALDH1A1 (0.63) ALDH1A1TSHRSLC6A3LMNADRD2
SCHEMBL9710602 0.88 ALDH1A1 (0.72) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL9181467 0.85 ALDH1A1 (0.58) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL11861506 0.83 ALDH1A1 (0.68) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL11867863 0.83 ALDH1A1 (0.68) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL9296560 0.82 ALDH1A1 (0.74) ALDH1A1TSHRSLC6A3KMT2AOPRL1
Hydrochloric Acid SCHEMBL11861149 0.82 ALDH1A1 (0.67) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL9297947 0.82 TSHR (0.73) ALDH1A1TSHRSLC6A3KMT2ALMNA
SCHEMBL11870408 0.81 ALDH1A1 (0.72) ALDH1A1TSHRSLC6A3KMT2ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512584-A 1,3,4-trisubstituted piperidine derivatives, the preparation and use thereof BASF AKTIENGESELLSCHAFT (DE) 1996-04-30 US disclosed
EP-0580644-B1 1,3,4-TRISUBSTITUTED PIPERIDINE DERIVATIVES, THEIR PRODUCTION AND USE BASF AG (DE) 1995-06-28 EP disclosed
EP-0580644-A1 1,3,4-TRISUBSTITUTED PIPERIDINE DERIVATIVES, THEIR PRODUCTION AND USE. BASF AG (DE) 1994-02-02 EP disclosed
WO-1992018480-A1 1,3,4-TRISUBSTITUTED PIPERIDINE DERIVATIVES, THEIR PRODUCTION AND USE BASF AKTIENGESELLSCHAFT (DE) 1992-10-29 WO disclosed