SCHEMBL8969833

SCHEMBL8969833

C=C1c2ccc(Cl)cc2N=C2CCCCCN12

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ACHE P22303 13/20 1.00
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
HDAC4 P56524 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970444 0.82 ACHE (0.70) ACHEKDM4EALDH1A1LMNAHTT
SCHEMBL8969901 0.79 ACHE (0.69) ACHEKDM4EALDH1A1HTTNPC1
SCHEMBL8968453 0.74 ACHE (1.00) ACHEALDH1A1LMNADRD2DRD4
SCHEMBL8968773 0.72 ACHE (0.97) ACHEALDH1A1LMNADRD2DRD4
SCHEMBL8968422 0.71 ACHE (1.00) ACHEALDH1A1LMNA
SCHEMBL8969321 0.70 ACHE (0.97) ACHEALDH1A1LMNA
SCHEMBL8969190 0.68 ACHE (0.89) ACHEALDH1A1LMNADRD2DRD4
SCHEMBL9382116 0.67 ACHE (0.52) ACHEKDM4EALDH1A1HTTSMN1; SMN2
SCHEMBL24330116 0.66 ACHE (0.67) ACHEKDM4EALDH1A1LMNAHTT
SCHEMBL9381904 0.66 ACHE (0.51) ACHEKDM4EALDH1A1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486512-A LEARNING ENHANCEMENT WARNER-LAMBERT COMPANY (US) 1996-01-23 US disclosed
EP-0597956-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1994-05-25 EP disclosed
WO-1993003034-A1 QUINAZOLINE DERIVATIVES AS ACETYLCHOLINESTERASE INHIBITORS WARNER-LAMBERT COMPANY (US) 1993-02-18 WO disclosed