SCHEMBL8970472

SCHEMBL8970472

CC(C)Oc1cccc(CC(=O)N(C)CC(OCC[N+]23CCC(c4ccccc4)(CC2)CC3)c2ccc(Cl)c(Cl)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 2/20 0.40
TACR1 P25103 2/20 0.39
TACR2 P21452 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8314434 0.88 CCR5 (0.48) CCR5TACR1TACR2
Hydrochloric Acid SCHEMBL8636368 0.87 CCR5 (0.47) CCR5TACR1TACR2
SCHEMBL9117577 0.87 CCR5 (0.39) CCR5TACR1TACR2
SCHEMBL8561473 0.82 TACR1 (0.42) CCR5TACR1
Hydrochloric Acid SCHEMBL8953818 0.80 CCR5 (0.37) CCR5TACR1TACR2
SCHEMBL8565799 0.80 TACR1 (0.40) CCR5TACR1
SCHEMBL8315849 0.74 TACR1 (0.43) CCR5TACR1TACR2
Hydrochloric Acid SCHEMBL8067085 0.74 TACR1 (0.48) CCR5TACR1TACR2
Hydrochloric Acid SCHEMBL8953619 0.74 TACR1 (0.42) CCR5TACR1TACR2
SCHEMBL8969597 0.72 TACR2 (0.53) TACR1TACR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700386-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1996-03-13 EP disclosed
WO-1995026338-A1 NEUROKININ RECEPTOR ANTAGONISTS SANOFI (FR) 1995-10-05 WO disclosed