SCHEMBL8971283

SCHEMBL8971283

COc1cc(N)c(Cl)cc1CC(=O)CC1CCN(CCNC(=O)N(C)C)CC1

nearest known ligand 0.49

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 14/20 0.49
MEN1 O00255 1/20 0.48
ALDH1A1 P00352 1/20 0.48
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 1/20 0.48
DRD2 P14416 1/20 0.47
DRD4 P21917 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8970723 0.86 HTR4 (0.55) HTR4MEN1ALDH1A1CYP3A4CYP2D6
SCHEMBL8971342 0.85 HTR4 (0.63) HTR4MEN1ALDH1A1CYP2D6CYP2C9
SCHEMBL8970664 0.85 HTR4 (0.67) HTR4MEN1ALDH1A1CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL8970748 0.84 HTR4 (0.62) HTR4MEN1ALDH1A1CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL6244982 0.84 HTR4 (0.66) HTR4MEN1ALDH1A1CYP3A4CYP2D6
SCHEMBL3230370 0.83 HTR4 (0.64) HTR4MEN1ALDH1A1CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8971374 0.83 DRD2 (0.52) HTR4MEN1ALDH1A1CYP2D6CYP2C9
SCHEMBL8970802 0.83 HTR4 (0.61) HTR4MEN1ALDH1A1CYP2D6CYP2C9
SCHEMBL8971324 0.83 HTR4 (0.60) HTR4MEN1ALDH1A1CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL8973729 0.82 HTR4 (0.63) HTR4MEN1ALDH1A1CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-A1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1996-03-13 EP disclosed