SCHEMBL8971494

SCHEMBL8971494

CCOP(=O)(CCC#N)C(F)F

nearest known ligand 0.36

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.36
TSHR P16473 3/20 0.35
PPARD Q03181 2/20 0.31
TP53 P04637 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
GAA P10253 1/20 0.30
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3842819 0.80 ACHE (0.35) ACHETSHRPPARDTP53TDP1
SCHEMBL9337737 0.77 ACHE (0.33) ACHETSHR
SCHEMBL9340199 0.76 ACHE (0.33) ACHETSHR
SCHEMBL9336312 0.76 ACHE (0.33) ACHETSHRPPARDMEN1KMT2A
SCHEMBL491513 0.74 TSHR (0.54) ACHETSHRPPARDTP53TDP1
SCHEMBL9337971 0.74 TSHR (0.38) ACHETSHR
SCHEMBL7790759 0.72 TSHR (0.41) ACHETSHRPPARDTP53TDP1
SCHEMBL8971372 0.72 CYP1A2 (0.44) TSHRPPARDMEN1KMT2A
SCHEMBL10343591 0.71 MEN1 (0.38) ACHETSHRMEN1KMT2A
SCHEMBL11726422 0.71 PPARD (0.57) ACHETSHRPPARDTP53TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5567840-A AS 4-AMINOBUTYRIC ACID AGONIST; MUSCLE RELAXANTS CIBA-GEIGY CORPORATION (US) 1996-10-22 US disclosed
US-5461040-A Therapy of spinal spacticity, multiple sclerosis, cerebral palsy, trigeminus neuralgia, drug withdrawal, pain CIBA-GEIGY CORPORATION (US) 1995-10-24 US disclosed
EP-0399949-B1 Substituted aminoalkylphosphinic acids CIBA GEIGY AG (CH) 1995-04-12 EP disclosed
US-5281747-A Pharmaceuticals CIBA-GEIGY CORPORATION (US) 1994-01-25 US disclosed
EP-0399949-A1 Substituted aminoalkylphosphinic acids CIBA-GEIGY AG (CH) 1990-11-28 EP disclosed