SCHEMBL8972034

SCHEMBL8972034

CCCCN1CCC(CC(=O)Cc2cc(Cl)c(N)cc2OCc2cc(OC)cc(OC)c2)CC1

nearest known ligand 0.69

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR4 Q13639 9/20 0.53
ACHE P22303 3/20 0.53
MEN1 O00255 2/20 0.53
ALDH1A1 P00352 2/20 0.53
CYP2D6 P10635 2/20 0.53
KMT2A Q03164 2/20 0.53
CYP2C9 P11712 1/20 0.53
TSHR P16473 1/20 0.53
TP53 P04637 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C19 P33261 1/20 0.52
DRD2 P14416 1/20 0.45
DRD4 P21917 1/20 0.45
CHRM4 P08173 1/20 0.42
CHRM5 P08912 1/20 0.42
ADRA2C P18825 1/20 0.42
CHRM3 P20309 1/20 0.42
HTR1D P28221 1/20 0.42
ADRA1B P35368 1/20 0.42
HTR2B P41595 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8971505 0.99 HTR4 (0.52) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL8971752 0.97 HTR4 (0.53) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8971733 0.90 MEN1 (0.52) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL8971284 0.89 MEN1 (0.57) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL3230370 0.88 HTR4 (0.64) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8973729 0.87 HTR4 (0.63) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL8971587 0.86 DRD2 (0.52) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8971867 0.85 DRD2 (0.51) HTR4ACHEMEN1ALDH1A1CYP2D6
SCHEMBL8971586 0.85 MEN1 (0.52) HTR4ACHEMEN1ALDH1A1CYP2D6
Hydrochloric Acid SCHEMBL8972032 0.84 MEN1 (0.51) HTR4ACHEMEN1ALDH1A1CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0700383-A1 NOVEL 1-PHENYLALKANONE 5-HT 4? RECEPTOR LIGANDS SYNTEX (U.S.A.) INC. (US) 1996-03-13 EP disclosed