SCHEMBL8972107

SCHEMBL8972107

CSc1ccccc1C1(C2c3cc(O)c(O)cc3CCN2C)CCC1

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MAOA P21397 1/20 0.44
DRD2 P14416 6/20 0.42
DRD3 P35462 1/20 0.42
DRD1 P21728 6/20 0.40
MAPK1 P28482 1/20 0.40
THPO P40225 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40
MTOR P42345 1/20 0.40
KDM4E B2RXH2 1/20 0.40
MAPT P10636 1/20 0.40
BLM P54132 1/20 0.40
PMP22 Q01453 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bromide SCHEMBL8747004 0.99 MAOA (0.43) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747048 0.85 MAOA (0.47) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747052 0.84 MAOA (0.46) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747172 0.84 DRD2 (0.54) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747167 0.84 MAOA (0.49) MAOADRD2DRD3DRD1MAPK1
Bromide SCHEMBL8747156 0.83 DRD2 (0.53) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747095 0.81 MAOA (0.43) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747168 0.81 DRD1 (0.44) MAOADRD2DRD3DRD1MAPK1
SCHEMBL8747006 0.81 MAOA (0.50) MAOADRD2DRD3DRD1MAPK1
Bromide SCHEMBL8747268 0.80 KDM4E (0.49) MAOADRD2DRD3DRD1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519034-A ANALGESICS THE BOOTS COMPANY PLC (GB) 1996-05-21 US disclosed
EP-0618900-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS. BOOTS CO PLC (GB) 1994-10-12 EP disclosed
WO-1993013073-A1 SUBSTITUTED TETRAHYDROISOQUINOLINES AND THEIR USE AS THERAPEUTIC AGENTS THE BOOTS COMPANY PLC (GB) 1993-07-08 WO disclosed