SCHEMBL8972309

SCHEMBL8972309

C/C=C/C1COC(c2ccc(-c3ccc(Cl)c(F)c3)cc2)OC1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 1/20 0.32
GRM2 Q14416 1/20 0.31
CYP11B1 P15538 3/20 0.31
CYP11B2 P19099 3/20 0.31
PGR P06401 1/20 0.31
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
PTGS1 P23219 1/20 0.30
PTGS2 P35354 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9311912 1.00 FFAR1 (0.32) FFAR1GRM2CYP11B1CYP11B2PGR
SCHEMBL8972300 1.00 FFAR1 (0.32) FFAR1GRM2CYP11B1CYP11B2PGR
SCHEMBL9311904 1.00 FFAR1 (0.32) FFAR1GRM2CYP11B1CYP11B2PGR
SCHEMBL8972495 0.88 AHR (0.39) PGRSLC6A2SLC6A4SLC6A3
SCHEMBL9312292 0.88 AHR (0.39) PGRSLC6A2SLC6A4SLC6A3
SCHEMBL8972500 0.88 AHR (0.39) PGRSLC6A2SLC6A4SLC6A3
SCHEMBL9312294 0.88 AHR (0.39) PGRSLC6A2SLC6A4SLC6A3
SCHEMBL8972512 0.88 CYP11B2 (0.33) CYP11B1CYP11B2PGR
SCHEMBL9312429 0.88 CYP11B2 (0.33) CYP11B1CYP11B2PGR
SCHEMBL9312426 0.88 CYP11B2 (0.33) CYP11B1CYP11B2PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0433836-B1 Halophenyl substituted dioxanes HOFFMANN LA ROCHE (CH) 1996-03-27 EP disclosed
US-5322638-A Halophenyl substituted dioxanes HOFFMANN-LA ROCHE INC. (US) 1994-06-21 US disclosed
EP-0433836-A2 Halophenyl substituted dioxanes F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed