SCHEMBL8973383

SCHEMBL8973383

N[C@]1(C(=O)O)C[C@H](C(=O)O)N(C(=O)Cc2ccccc2)C1

nearest known ligand 0.64

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GRM6 O15303 1/20 0.64
GRM2 Q14416 8/20 0.61
GRM3 Q14832 5/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973200 0.87 GRM2 (0.65) GRM6GRM2GRM3
SCHEMBL8972828 0.82 GRM2 (0.65) GRM6GRM2GRM3
SCHEMBL8973083 0.79 GRM2 (0.58) GRM6GRM2GRM3
SCHEMBL5566850 0.78 GRM2 (0.57) GRM6GRM2GRM3
SCHEMBL4665515 0.78 GRM2 (0.57) GRM6GRM2GRM3
SCHEMBL5567277 0.78 GRM2 (0.57) GRM6GRM2GRM3
SCHEMBL4665462 0.78 GRM2 (0.57) GRM6GRM2GRM3
SCHEMBL5567611 0.78 GRM2 (0.57) GRM6GRM2GRM3
SCHEMBL8061968 0.78 GRM6 (1.00) GRM6GRM2GRM3
SCHEMBL8973264 0.78 GRM6 (1.00) GRM6GRM2GRM3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0703218-A1 Pyrrolidinyl di-carboxylic acid derivatives as metabotropic glutamate receptor antagonists ELI LILLY AND COMPANY (US) 1996-03-27 EP disclosed
WO-1996005828-A1 PYRROLIDINYL DI-CARBOXYLIC ACID DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-02-29 WO disclosed