SCHEMBL8973617

SCHEMBL8973617

O=C1CN(S(=O)(=O)c2cc3ccc(Cl)cc3cc2Cl)C(=S)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 2/20 0.41
USP2 O75604 1/20 0.39
ALDH1A1 P00352 1/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 1/20 0.39
TSHR P16473 4/20 0.38
L3MBTL1 Q9Y468 2/20 0.38
ALOX15 P16050 1/20 0.38
ATM Q13315 1/20 0.36
PIM1 P11309 1/20 0.34
HTT P42858 2/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
LMNA P02545 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TRPV4 Q9HBA0 1/20 0.33
CMA1 P23946 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
CNR1 P21554 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8973450 0.89 PKM (0.44) PKMUSP2ALDH1A1MEN1KMT2A
SCHEMBL8789825 0.86 PKM (0.56) PKMUSP2ALDH1A1MEN1KMT2A
SCHEMBL8973740 0.77 MEN1 (0.48) PKMUSP2ALDH1A1MEN1KMT2A
SCHEMBL8789027 0.73 PKM (0.59) PKMUSP2ALDH1A1MEN1KMT2A
SCHEMBL8973564 0.72 MEN1 (0.38) ALDH1A1MEN1KMT2APOLBHSD17B10
SCHEMBL8973357 0.71 MEN1 (0.51) ALDH1A1MEN1KMT2APOLBGAA
SCHEMBL10672409 0.71 KMT2A (0.51) ALDH1A1MEN1KMT2APOLBTSHR
SCHEMBL8973126 0.70 MEN1 (0.50) ALDH1A1MEN1KMT2APOLBGAA
SCHEMBL8799304 0.70 MEN1 (0.32) MEN1KMT2APOLBTDP1
SCHEMBL7051174 0.68 PKM (0.46) PKMMEN1KMT2APOLBTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE35279-E ALDOSE REDUCTASE INHIBITORS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1996-06-18 US disclosed
US-5202339-A Hypoglycemic, hypolipedemic agents MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1993-04-13 US disclosed
EP-0305947-B1 HYDANTOIN DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THE SAME AS WELL AS THEIR USE MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1992-07-29 EP disclosed
US-5004751-A Antidiabetic agents; aldoe reductase inhibitors MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1991-04-02 US disclosed
US-4914099-A TREATMENT OR PREVENTION OF DIABETIC COMPLICATIONS MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1990-04-03 US disclosed
WO-1989001934-A1 HYDANTOIN DERIVATIVES MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-09 WO disclosed
EP-0305947-A1 Hydantoin derivatives, process for their preparation and pharmaceutical compositions containing the same as well as their use MOCHIDA PHARMACEUTICAL CO., LTD. (JP) 1989-03-08 EP disclosed