SCHEMBL8974171

SCHEMBL8974171

CS(=O)(=O)c1ccc(C2=CC(C(F)(F)F)(C(F)(F)F)C=C2c2ccncc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 13/20 0.48
PTGS1 P23219 2/20 0.48
MAPK11 Q15759 2/20 0.42
MAPK14 Q16539 2/20 0.42
MAPK13 O15264 1/20 0.42
RAF1 P04049 1/20 0.42
MAPK9 P45984 1/20 0.42
MAPK12 P53778 1/20 0.42
ALDH1A1 P00352 1/20 0.42
ALOX5 P09917 1/20 0.42
CSNK1A1 P48729 1/20 0.42
CSNK1D P48730 1/20 0.42
CSNK1E P49674 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
CSNK1A1L Q8N752 1/20 0.42
MELK Q14680 1/20 0.42
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
SCD O00767 1/20 0.39
KIF11 P52732 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974655 0.87 PTGS2 (0.56) PTGS2PTGS1KIF11
SCHEMBL8974490 0.85 CA2 (0.50) PTGS2PTGS1ALOX5KIF11
SCHEMBL8973922 0.85 PTGS2 (0.66) PTGS2PTGS1
SCHEMBL8975150 0.84 PTGS2 (0.51) PTGS2PTGS1
SCHEMBL8974513 0.83 PTGS2 (0.51) PTGS2PTGS1MAPK11MAPK14MAPK13
SCHEMBL8974291 0.82 KCNH2 (0.53) PTGS2PTGS1KIF11
SCHEMBL8974078 0.81 PTGS2 (0.49) PTGS2PTGS1MAPK11MAPK14MAPK13
SCHEMBL8974501 0.81 PTGS2 (0.47) PTGS2PTGS1KIF11
SCHEMBL8974098 0.79 PTGS2 (0.48) PTGS2PTGS1MAPK11MAPK14MAPK13
SCHEMBL9116419 0.79 PTGS2 (0.70) PTGS2PTGS1MAPK11MAPK14MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed