SCHEMBL8974263

SCHEMBL8974263

CC1C=C(c2ccc(S(C)(=O)=O)cc2)C(c2ccc(C(F)(F)F)cn2)=C1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.45
GPR119 Q8TDV5 1/20 0.44
KIF11 P52732 1/20 0.43
PTGS1 P23219 4/20 0.42
IDO1 P14902 2/20 0.40
TDO2 P48775 1/20 0.40
KCNH2 Q12809 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974815 0.93 PTGS2 (0.44) PTGS2KIF11PTGS1IDO1TDO2
SCHEMBL8974463 0.90 KIF11 (0.46) PTGS2GPR119KIF11PTGS1IDO1
SCHEMBL8974487 0.89 KIF11 (0.50) PTGS2KIF11PTGS1
SCHEMBL8974797 0.89 PTGS2 (0.44) PTGS2GPR119KIF11PTGS1IDO1
SCHEMBL8974779 0.87 PTGS2 (0.45) PTGS2GPR119KIF11PTGS1
SCHEMBL8974330 0.87 PTGS2 (0.45) PTGS2GPR119KIF11PTGS1IDO1
SCHEMBL8974329 0.86 PTGS2 (0.47) PTGS2GPR119KIF11PTGS1IDO1
SCHEMBL8974238 0.86 PTGS2 (0.46) PTGS2GPR119KIF11PTGS1
SCHEMBL8974307 0.86 PTGS2 (0.57) PTGS2KIF11PTGS1
SCHEMBL8974632 0.84 KIF11 (0.50) PTGS2KIF11PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed