SCHEMBL8974295

SCHEMBL8974295

NS(=O)(=O)c1ccc(C2=CC(C(F)(F)F)C=C2c2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 9/20 0.43
CA1 P00915 3/20 0.39
CA2 P00918 3/20 0.39
CA9 Q16790 2/20 0.39
CA12 O43570 1/20 0.39
CA4 P22748 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39
PTGS2 P35354 5/20 0.37
PTGS1 P23219 2/20 0.37
ALOX5AP P20292 1/20 0.37
FEN1 P39748 1/20 0.37
CYP2C9 P11712 1/20 0.34
COMT P21964 1/20 0.34
PDPK1 O15530 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974346 0.88 CA1 (0.40) KIF11CA1CA2CA9CA12
SCHEMBL8974593 0.87 KIF11 (0.38) KIF11PTGS2ALOX5APFEN1
SCHEMBL8973842 0.87 KIF11 (0.43) KIF11CA1CA2CA9CA12
SCHEMBL9118202 0.85 PPARD (0.39) KIF11
SCHEMBL8974834 0.85 KIF11 (0.41) KIF11CA1CA2CA9CA12
SCHEMBL8974190 0.84 KIF11 (0.40) KIF11CA1CA2CA9CA12
SCHEMBL8974163 0.84 KIF11 (0.40) KIF11CA1CA2CA9CA12
SCHEMBL8974154 0.84 KIF11 (0.40) KIF11CA1CA2CA9CA12
SCHEMBL6260512 0.82 KIF11 (0.59) KIF11CA1CA2CA9CA12
SCHEMBL8974062 0.82 KIF11 (0.45) KIF11CA1CA2CA9CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed