SCHEMBL8974154

SCHEMBL8974154

NS(=O)(=O)c1ccc(C2=CC(C(=O)O)C=C2c2ccc(C(F)(F)F)cc2)cn1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 7/20 0.40
PPARD Q03181 3/20 0.38
MAP4K4 O95819 1/20 0.38
CA12 O43570 3/20 0.36
CA1 P00915 3/20 0.36
CA2 P00918 3/20 0.36
CA9 Q16790 3/20 0.36
CA4 P22748 1/20 0.36
CA6 P23280 1/20 0.36
CA5A P35218 1/20 0.36
CA7 P43166 1/20 0.36
CA13 Q8N1Q1 1/20 0.36
CA14 Q9ULX7 1/20 0.36
ALOX5AP P20292 1/20 0.35
FEN1 P39748 1/20 0.35
PTGS1 P23219 2/20 0.35
PTGS2 P35354 2/20 0.35
MAPT P10636 1/20 0.35
POLB P06746 1/20 0.35
COMT P21964 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974707 0.88 PPARD (0.38) KIF11PPARDMAP4K4ALOX5APFEN1
SCHEMBL8974506 0.86 CA1 (0.44) MAP4K4CA12CA1CA2CA9
SCHEMBL8974153 0.86 KIF11 (0.40) KIF11PPARDCA12CA1CA2
SCHEMBL8973842 0.84 KIF11 (0.43) KIF11CA12CA1CA2CA9
SCHEMBL8974295 0.84 KIF11 (0.43) KIF11CA12CA1CA2CA9
SCHEMBL8974190 0.83 KIF11 (0.40) KIF11PPARDMAP4K4CA12CA1
SCHEMBL8974090 0.82 KIF11 (0.62) KIF11CA12CA1CA2CA9
SCHEMBL8974834 0.82 KIF11 (0.41) KIF11PPARDCA12CA1CA2
SCHEMBL8974163 0.81 KIF11 (0.40) KIF11PPARDCA12CA1CA2
SCHEMBL8973844 0.81 KIF11 (0.40) KIF11PPARDMAP4K4CA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed