SCHEMBL8974406

SCHEMBL8974406

NS(=O)(=O)c1ccc(C2=CCC=C2c2ccc(F)cc2)cc1

nearest known ligand 0.60

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 14/20 0.60
PTGS1 P23219 11/20 0.60
MAOA P21397 1/20 0.54
MAOB P27338 1/20 0.54
SOS1 Q07889 1/20 0.53
CA2 P00918 5/20 0.52
CA12 O43570 2/20 0.52
CA9 Q16790 2/20 0.52
CA1 P00915 3/20 0.49
CA4 P22748 2/20 0.49
CA7 P43166 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9118818 0.84 PTGS2 (0.48) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974157 0.84 CA2 (0.45) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974436 0.84 CA2 (0.45) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974782 0.84 CA2 (0.68) PTGS2PTGS1MAOAMAOBCA2
SCHEMBL8974243 0.84 CA2 (0.71) PTGS2PTGS1CA2CA12CA9
SCHEMBL8974557 0.83 PTGS2 (0.60) PTGS2PTGS1SOS1CA2CA12
SCHEMBL1430142 0.82 CA2 (0.76) PTGS2PTGS1MAOAMAOBSOS1
SCHEMBL8973815 0.82 CA2 (0.52) PTGS2PTGS1CA2CA12CA9
SCHEMBL8974305 0.82 CA2 (0.64) PTGS2PTGS1CA2CA12CA9
SCHEMBL8974750 0.82 CA2 (0.64) PTGS2PTGS1MAOAMAOBCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO claimed
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
WO-1995030656-A1 SUBSTITUTED CYCLOPENTADIENYL COMPOUNDS FOR THE TREATMENT OF INFLAMMATION G.D. SEARLE & CO. (US) 1995-11-16 WO disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed