SCHEMBL8974476

SCHEMBL8974476

O=C(O)c1ccccc1N(S(=O)(=O)c1ccccc1)S(=O)(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
ALOX15 P16050 1/20 0.46
CYP3A4 P08684 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
APOBEC3G Q9HC16 1/20 0.44
KMT2A Q03164 2/20 0.43
HSD11B1 P28845 1/20 0.43
KEAP1 Q14145 1/20 0.42
NFE2L2 Q16236 1/20 0.42
GAA P10253 3/20 0.42
NPSR1 Q6W5P4 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
ATM Q13315 1/20 0.41
CA1 P00915 2/20 0.41
CA2 P00918 2/20 0.41
KDM4E B2RXH2 1/20 0.41
CA12 O43570 1/20 0.41
HMGB1 P09429 1/20 0.41
HPGD P15428 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974735 0.82 MCL1 (0.50) ALDH1A1KMT2ATDP1
SCHEMBL2556706 0.79 ALDH1A1 (0.48) ALDH1A1ALOX15KMT2AGAACA1
SCHEMBL18158039 0.74 ALDH1A1 (0.56) ALDH1A1ALOX15GAATDP1CA1
SCHEMBL13066508 0.73 ALDH1A1 (0.62) ALDH1A1ALOX15GAACA1CA2
SCHEMBL16550141 0.73 APOBEC3G (0.52) ALDH1A1CYP3A4CYP2C9CYP2C19APOBEC3G
SCHEMBL5853971 0.73 CYP3A4 (0.47) ALDH1A1CYP3A4CYP2C9CYP2C19APOBEC3G
SCHEMBL5853978 0.73 TEAD1 (0.49) ALDH1A1CYP3A4CYP2C9CYP2C19APOBEC3G
SCHEMBL2776583 0.71 ALDH1A1 (0.59) ALDH1A1ALOX15GAACA1CA2
SCHEMBL14150723 0.71 ALDH1A1 (0.52) ALDH1A1ALOX15GAACA1CA2
SCHEMBL7195145 0.71 ALDH1A1 (0.52) ALDH1A1ALOX15CYP3A4CYP2C9GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996039132-A1 N,N-DISULFONYLATED AMINOBENZENE CARBOXYLIC ACIDS AND THE USE THEREOF AS THROMBIN INHIBITORS 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1996-12-12 WO disclosed
US-5559150-A ANTICOAGULANT, ANTITUMOR, ANTIINFLAMMATORY 3-DIMENSIONAL PHARMACEUTICALS, INC. (US) 1996-09-24 US disclosed