SCHEMBL8974489

SCHEMBL8974489

COCOc1c(OC)cc(CO[Si](C)(C)C(C)(C)C)c2cccc(C)c12

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 1/20 0.35
ABCC1 P33527 1/20 0.35
ABCG2 Q9UNQ0 1/20 0.35
PTPN1 P18031 1/20 0.34
HTR1A P08908 1/20 0.31
ADRA1D P25100 1/20 0.31
ADRA1A P35348 1/20 0.31
ADRA1B P35368 1/20 0.31
NFKB1 P19838 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974383 0.84 BACE1 (0.33) PTPN1
SCHEMBL8974210 0.82 PTPN1 (0.32) PTPN1
SCHEMBL8974794 0.80 PTPN1 (0.44) ABCB1ABCC1ABCG2PTPN1
SCHEMBL8974503 0.74 ABCB1 (0.37) ABCB1ABCC1ABCG2HTR1AADRA1D
SCHEMBL8974218 0.72 BACE1 (0.34)
SCHEMBL8974498 0.72 MAOA (0.31)
SCHEMBL8973931 0.71 PTPN1 (0.42) PTPN1
SCHEMBL9900805 0.69 PREP (0.34)
SCHEMBL29437982 0.69 PREP (0.34)
SCHEMBL3151669 0.67 F2RL3 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527948-A SUBSTITUTED NAPHTHYL-ALKENOIC ACIDS FOR TREATING AUTOIMMUNE DISORDERS EISAI CORP. LTD. (JP) 1996-06-18 US disclosed
US-5298649-A Antiinflammatory agents, rheumatic agents and treatment of autoimmune diseases EISAI CO., LTD. (JP) 1994-03-29 US disclosed
EP-0376288-B1 Naphthalene derivative EISAI CO LTD (JP) 1994-03-09 EP disclosed
US-5134111-A Inhibitors of interleukin-1 as antiinflammatory agents EISAI CO., LTD. (JP) 1992-07-28 US disclosed
EP-0376288-A1 Naphthalene derivative Eisai Co., Ltd. (JP) 1990-07-04 EP disclosed