SCHEMBL8974582

SCHEMBL8974582

CS(=O)(=O)c1ccc(C2=CC(CO)(CO)C=C2c2ccncc2)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 12/20 0.48
PTGS1 P23219 4/20 0.48
MAPK13 O15264 2/20 0.45
MAPK12 P53778 2/20 0.45
MAPK11 Q15759 2/20 0.45
MAPK14 Q16539 2/20 0.45
RAF1 P04049 1/20 0.45
MAPK9 P45984 1/20 0.45
SLC22A12 Q96S37 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2C9 P11712 1/20 0.42
MELK Q14680 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974089 0.87 PTGS2 (0.46) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL8974325 0.85 CA2 (0.50) PTGS2PTGS1SLC22A12
SCHEMBL8974098 0.85 PTGS2 (0.48) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL8974066 0.84 PTGS2 (0.64) PTGS2PTGS1CYP3A4CYP2C9
SCHEMBL8974391 0.84 PTGS2 (0.59) PTGS2PTGS1
SCHEMBL8974536 0.83 PTGS2 (0.52) PTGS2PTGS1
SCHEMBL8974078 0.81 PTGS2 (0.49) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL8974513 0.80 PTGS2 (0.51) PTGS2PTGS1MAPK13MAPK12MAPK11
SCHEMBL8974812 0.80 PTGS2 (0.49) PTGS2PTGS1
SCHEMBL9116419 0.79 PTGS2 (0.70) PTGS2PTGS1MAPK13MAPK12MAPK11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5576339-A Pyridyl substituted cyclopentadienes for the treatment of inflamation HUANG HORNG-CHIH (US) 1996-11-19 US disclosed
US-5418254-A Side effect reduction G. D. SEARLE & CO. (US) 1995-05-23 US disclosed