SCHEMBL8974767

SCHEMBL8974767

Cc1cc(-c2c(-c3ccc(S(C)(=O)=O)cc3)n[nH]c2C(F)(F)F)ccc1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRB P28702 2/20 0.44
RXRA P19793 1/20 0.44
LRRK2 Q5S007 2/20 0.43
NR1H2 P55055 1/20 0.39
PTGS2 P35354 5/20 0.39
PTGDR2 Q9Y5Y4 1/20 0.39
PTGS1 P23219 2/20 0.38
MAPK1 P28482 2/20 0.38
MAP2K4 P45985 2/20 0.38
MAPK6 Q16659 2/20 0.38
MAPKAPK3 Q16644 1/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
CNR1 P21554 1/20 0.38
NR2F2 P24468 1/20 0.38
CNR2 P34972 1/20 0.38
KMT2A Q03164 1/20 0.38
GPR55 Q9Y2T6 1/20 0.38
MAPKAPK5 Q8IW41 1/20 0.38
CA12 O43570 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8975131 0.91 LRRK2 (0.52) RXRBRXRALRRK2PTGS2MAP2K4
SCHEMBL7777889 0.87 PTGS2 (0.49) LRRK2NR1H2PTGS2PTGS1
SCHEMBL7778114 0.85 LRRK2 (0.47) LRRK2PTGS2PTGDR2PTGS1MAPK1
SCHEMBL7780442 0.82 PTGS2 (0.51) LRRK2NR1H2PTGS2PTGS1GYS1
SCHEMBL7780652 0.82 PTGS2 (0.53) LRRK2NR1H2PTGS2PTGS1MAPT
SCHEMBL7772850 0.81 PTGS2 (0.51) LRRK2NR1H2PTGS2PTGDR2PTGS1
SCHEMBL7779584 0.81 PTGS2 (0.58) LRRK2PTGS2PTGS1MEN1MAPT
SCHEMBL7779772 0.81 LRRK2 (0.50) LRRK2PTGS2PTGS1
SCHEMBL7779920 0.80 LRRK2 (0.53) LRRK2NR1H2PTGS2PTGS1
SCHEMBL7780827 0.80 LRRK2 (0.48) LRRK2PTGS2MAPK1MAP2K4MAPK6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486534-A 3,4-substituted pyrazoles for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-01-23 US disclosed