SCHEMBL8975131

SCHEMBL8975131

Cc1cc(-c2c(-c3ccc(S(N)(=O)=O)cc3)n[nH]c2C(F)(F)F)ccc1C(=O)O

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 10/20 0.52
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
MAP2K7 O14733 1/20 0.41
MAP2K4 P45985 1/20 0.41
PTGS2 P35354 1/20 0.40
MAPT P10636 3/20 0.39
GPR55 Q9Y2T6 3/20 0.39
CNR1 P21554 2/20 0.39
CNR2 P34972 2/20 0.39
MEN1 O00255 1/20 0.39
NR2F2 P24468 1/20 0.39
KMT2A Q03164 1/20 0.39
CA12 O43570 2/20 0.39
CA9 Q16790 2/20 0.39
ALDH1A1 P00352 1/20 0.39
BLM P54132 1/20 0.39
GYS1 P13807 2/20 0.39
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974767 0.91 RXRB (0.44) LRRK2RXRARXRBMAP2K4PTGS2
SCHEMBL7780622 0.87 LRRK2 (0.57) LRRK2MAP2K7MAP2K4PTGS2GYS1
SCHEMBL7779735 0.85 LRRK2 (0.57) LRRK2MAP2K7MAP2K4PTGS2MAPT
SCHEMBL7777855 0.83 LRRK2 (0.55) LRRK2MAP2K7MAP2K4PTGS2GYS1
SCHEMBL7780114 0.82 PTGS2 (0.54) LRRK2PTGS2MAPTGPR55CNR1
SCHEMBL7777620 0.81 LRRK2 (0.60) LRRK2MAP2K7MAP2K4PTGS2CA12
SCHEMBL7777532 0.81 LRRK2 (0.53) LRRK2MAP2K7MAP2K4PTGS2MAPT
SCHEMBL7779616 0.81 LRRK2 (0.64) LRRK2MAP2K7MAP2K4PTGS2CA1
SCHEMBL7773326 0.80 LRRK2 (0.68) LRRK2MAP2K7MAP2K4PTGS2MAPT
SCHEMBL7780655 0.79 CA12 (0.57) LRRK2MAP2K4PTGS2MAPTGPR55

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5486534-A 3,4-substituted pyrazoles for the treatment of inflammation G. D. SEARLE & CO. (US) 1996-01-23 US disclosed