SCHEMBL8975149

SCHEMBL8975149

Clc1ccc2c(NCCc3ccccc3)ncnc2c1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 5/20 0.71
MAPK1 P28482 3/20 0.70
LMNA P02545 3/20 0.70
EGFR P00533 1/20 0.70
APP P05067 1/20 0.70
PIK3CD O00329 2/20 0.69
PIK3R1 P27986 2/20 0.69
CNR1 P21554 1/20 0.69
CNR2 P34972 1/20 0.69
NR2F2 P24468 1/20 0.62
KDM4E B2RXH2 1/20 0.60
ALDH1A1 P00352 1/20 0.60
HPGD P15428 1/20 0.60
PPARG P37231 1/20 0.58
RXFP1 Q9HBX9 1/20 0.58
NR2E3 Q9Y5X4 1/20 0.58
NCOR2 Q9Y618 1/20 0.58
CCNC P24863 1/20 0.57
CDKN1A P38936 1/20 0.57
CDK8 P49336 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9921509 0.89 PIK3CD (0.85) HTTMAPK1LMNAEGFRAPP
SCHEMBL8548141 0.87 MAPK1 (0.62) HTTMAPK1LMNAEGFRAPP
SCHEMBL11846406 0.85 KDM4E (0.63) HTTMAPK1LMNAPIK3CDPIK3R1
SCHEMBL8540683 0.85 HTT (0.65) HTTMAPK1LMNAEGFRAPP
SCHEMBL3979500 0.83 KDM4E (0.77) HTTMAPK1LMNAPIK3CDPIK3R1
SCHEMBL8497590 0.83 APP (1.00) HTTMAPK1LMNAEGFRAPP
SCHEMBL8541525 0.82 HTT (0.81) HTTMAPK1LMNAEGFRAPP
SCHEMBL17557570 0.82 CNR1 (1.00) HTTMAPK1LMNAEGFRAPP
SCHEMBL9921357 0.82 PIK3CD (1.00) HTTMAPK1LMNAEGFRAPP
SCHEMBL11855329 0.81 HDAC1 (0.60) HTTMAPK1LMNAPIK3CDPIK3R1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705253-A1 ARALKYLAMINOQUINAZOLINES BAYER AG (DE) 1996-04-10 EP claimed
WO-1995000496-A1 ARALKYLAMINOQUINAZOLINES BAYER AKTIENGESELLSCHAFT (DE) 1995-01-05 WO claimed
EP-0705253-A1 ARALKYLAMINOQUINAZOLINES BAYER AG (DE) 1996-04-10 EP disclosed
WO-1995000496-A1 ARALKYLAMINOQUINAZOLINES BAYER AKTIENGESELLSCHAFT (DE) 1995-01-05 WO disclosed