SCHEMBL8975446

SCHEMBL8975446

CC(COc1ccc(CC2SC(=O)NC2=O)cc1)NCC(O)CN(C)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARG P37231 13/20 0.50
FFAR1 O14842 8/20 0.49
RARG P13631 1/20 0.47
RXRA P19793 1/20 0.47
PPARA Q07869 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8974677 0.88 PPARG (0.57) PPARGFFAR1PPARA
SCHEMBL8974649 0.86 FFAR1 (0.53) PPARGFFAR1PPARA
SCHEMBL8974734 0.85 FFAR1 (0.56) PPARGFFAR1PPARA
SCHEMBL8975130 0.84 FFAR1 (0.52) PPARGFFAR1PPARA
SCHEMBL8974731 0.83 FFAR1 (0.50) PPARGFFAR1PPARA
SCHEMBL8974550 0.82 FFAR1 (0.52) PPARGFFAR1RXRA
SCHEMBL8974743 0.82 FFAR1 (0.59) PPARGFFAR1PPARA
SCHEMBL8975029 0.81 FFAR1 (0.50) PPARGFFAR1RXRA
SCHEMBL8974598 0.80 FFAR1 (0.49) PPARGFFAR1RXRA
SCHEMBL8974608 0.80 FFAR1 (0.54) PPARGFFAR1PPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5578620-A TREATMENT OF DIABETES AND HYPERLIPEMIA SANKYO COMPANY, LIMITED (JP) 1996-11-26 US disclosed
EP-0678511-A2 Thiazolidine and oxazolidine derivatives, their preparation and their medical use SANKYO COMPANY LIMITED (JP) 1995-10-25 EP disclosed