SCHEMBL8976576

SCHEMBL8976576

CCOP(=O)(Cc1ccccc1)CC(O)CCl

nearest known ligand 0.44

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.44
MAPK1 P28482 2/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
NR1I2 O75469 1/20 0.40
GAA P10253 2/20 0.40
TSHR P16473 3/20 0.39
NPSR1 Q6W5P4 2/20 0.38
HPGD P15428 2/20 0.38
ALOX15 P16050 1/20 0.38
KMT2A Q03164 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.36
KCNH2 Q12809 1/20 0.36
MEN1 O00255 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8751389 1.00 POLB (0.44) POLBMAPK1ALDH1A1MAPTNR1I2
SCHEMBL8814946 0.89 LTA4H (0.44) CYP2C19
SCHEMBL8815671 0.87 POLB (0.35) POLBMAPK1ALDH1A1MAPTGAA
SCHEMBL563856 0.79 NPSR1 (0.50) POLBNR1I2TSHRNPSR1HPGD
SCHEMBL340010 0.78 POLB (0.42) POLBMAPK1ALDH1A1MAPTNR1I2
SCHEMBL9063192 0.78 MEN1 (0.45) ALDH1A1MAPTGAAKMT2ASMN1; SMN2
SCHEMBL9063188 0.78 MEN1 (0.45) ALDH1A1MAPTGAAKMT2ASMN1; SMN2
Hydrogen Peroxide SCHEMBL8609520 0.78 POLB (0.46) POLBNR1I2TSHRNPSR1HPGD
SCHEMBL5417880 0.76 NPSR1 (0.47) POLBNR1I2TSHRNPSR1HPGD
SCHEMBL7617120 0.73 FOLH1 (0.63)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5545631-A GAMMA-AMINOBUTYRIC ACID ANTAGONIST; TREATS PETIT-MAL TYPE EPILEPSIES CIBA-GEIGY CORPORATION (US) 1996-08-13 US disclosed
US-5500418-A ANTIEPILEPTIC CIBA-GEIGY CORPORATION (US) 1996-03-19 US disclosed
US-5407922-A GABA antagonists CIBA-GEIGY CORPORATION (US) 1995-04-18 US disclosed
US-5376684-A Aminobutyric acid antagonist; antiepileptic agent CIBA-GEIGY CORPORATION (US) 1994-12-27 US disclosed
US-5229379-A Gamma-aminobutyric acid antagonists CIBA-GEIGY CORPORATION (US) 1993-07-20 US disclosed