SCHEMBL8976704

SCHEMBL8976704

COc1cc2ncnc(Nc3nccc4ccccc34)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
EGFR P00533 16/20 1.00
KDR P35968 4/20 0.66
RET P07949 3/20 0.66
LCK P06239 3/20 0.64
KRAS P01116 1/20 0.61
SOS1 Q07889 1/20 0.61
FLT1 P17948 1/20 0.60
CLK1 P49759 1/20 0.59
ABCG2 Q9UNQ0 1/20 0.59
RIPK2 O43353 1/20 0.58
EPHB2 P29323 1/20 0.58
ATM Q13315 1/20 0.58
SRC P12931 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6180170 0.85 EGFR (0.76) EGFRKDRRETLCKFLT1
Hydrochloric Acid SCHEMBL6180124 0.84 EGFR (0.74) EGFRKDRRETLCKFLT1
SCHEMBL8976474 0.80 EGFR (0.66) EGFRKDRRETFLT1
SCHEMBL1257431 0.80 EGFR (1.00) EGFRKDRRETLCKFLT1
SCHEMBL29515328 0.80 EGFR (1.00) EGFRKDRRETLCKFLT1
SCHEMBL6181200 0.80 EGFR (0.74) EGFRKDRRETLCKFLT1
SCHEMBL7120134 0.80 RET (0.71) EGFRKDRRETLCKFLT1
Hydrochloric Acid SCHEMBL5475737 0.79 EGFR (1.00) EGFRKDRRETLCKRIPK2
Hydrochloric Acid SCHEMBL6180787 0.79 EGFR (0.74) EGFRKDRRETLCKCLK1
SCHEMBL8976742 0.79 EGFR (0.74) EGFRKDRRETLCKFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5580870-A ANTICARCINOGENIC AGENTS ZENECA LIMITED (GB) 1996-12-03 US disclosed
EP-0602851-B1 Quinazoline derivatives ZENECA LTD (GB) 1996-10-09 EP disclosed
EP-0602851-A1 Quinazoline derivatives ZENECA LIMITED (GB) 1994-06-22 EP disclosed