SCHEMBL8978393

SCHEMBL8978393

O=c1cc[nH]c(=O)n1NC=Cc1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.36
NPC1 O15118 2/20 0.36
ALDH1A1 P00352 5/20 0.35
LMNA P02545 2/20 0.35
MAPK1 P28482 2/20 0.35
TRPA1 O75762 1/20 0.35
ALOX5 P09917 1/20 0.35
ELANE P08246 1/20 0.35
DPYD Q12882 1/20 0.33
CCNE1 P24864 1/20 0.33
CDK2 P24941 1/20 0.33
KDM4E B2RXH2 4/20 0.33
THRB P10828 1/20 0.33
HPGD P15428 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 2/20 0.32
MAPT P10636 2/20 0.32
KMT2A Q03164 2/20 0.32
POLB P06746 1/20 0.32
PKM P14618 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4445914 0.71 CYP1A2 (0.44) ALDH1A1LMNAMAPK1HPGDMAPT
SCHEMBL8978389 0.67 CRBN (0.50) RAB9ANPC1ALDH1A1LMNAMAPK1
SCHEMBL8978384 0.67 CRBN (0.50) RAB9ANPC1ALDH1A1LMNAMAPK1
SCHEMBL27701056 0.66 BRD4 (0.33) KDM4E
SCHEMBL2181559 0.66
Benzaldehyde SCHEMBL27944564 0.65 CYP2A6 (0.47) ALDH1A1LMNAMAPK1TRPA1ALOX5
SCHEMBL9277794 0.64
SCHEMBL45000 0.61 GSK3A (0.54) RAB9ANPC1ALDH1A1LMNAMAPK1
SCHEMBL991992 0.61 NPC1 (0.52) RAB9ANPC1ALDH1A1LMNAMAPK1
SCHEMBL2561874 0.60 CYP2A6 (0.31)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705265-A1 NOVEL CHEMICAL COMPOUNDS HAVING PDE-IV INHIBITION ACTIVITY Euroceltique S.A. (LU) 1996-04-10 EP disclosed