SCHEMBL8979642

SCHEMBL8979642

CN(C(=O)CCCl)c1ccccc1F

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.42
TP53 P04637 2/20 0.42
TSHR P16473 1/20 0.42
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41
GPBAR1 Q8TDU6 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.38
POLB P06746 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAPK1 P28482 1/20 0.36
GAA P10253 1/20 0.36
KDM4E B2RXH2 1/20 0.36
LMNA P02545 1/20 0.35
ALOX15 P16050 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
ESR1 P03372 1/20 0.35
TACR1 P25103 1/20 0.35
OPRM1 P35372 1/20 0.34
KCNH2 Q12809 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23723512 0.86 ALDH1A1 (0.43) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL10272367 0.85 ALDH1A1 (0.48) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL31287485 0.82 ALDH1A1 (0.44) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL13684202 0.81 ALDH1A1 (0.47) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL11339370 0.81 ALDH1A1 (0.44) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL4128007 0.80 CES2 (0.43) ALDH1A1TP53TSHR
SCHEMBL1114942 0.80 HDAC3 (0.44) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL12679952 0.80 ALDH1A1 (0.40) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL1115146 0.80 HDAC3 (0.44) ALDH1A1TP53TSHRDDB1CRBN
SCHEMBL31606582 0.79 ALDH1A1 (0.43) ALDH1A1TP53TSHRDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5512594-A ADMINISTERING TO TREAT A MEDICAL CONDITION MEDIATED BY ONE OR MORE LEUKOTRIENES ZENECA LIMITED (GB) 1996-04-30 US disclosed
WO-1994025453-A1 4-ARYL-4-HYDROXY-TETRAHYDROPYRANS AND 3-ARYL-3-HYDROXY-TETRAHYDROFURANS AS 5-LIPOXYGENASE INHIBITORS ZENECA LIMITED (GB) 1994-11-10 WO disclosed