SCHEMBL8979697

SCHEMBL8979697

CCCC[Sn](CCCC)(CCCC)c1ccc(C(N)=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK1 P28482 2/20 0.46
KMT2A Q03164 2/20 0.46
MEN1 O00255 1/20 0.46
APAF1 O14727 1/20 0.46
RGS12 O14924 1/20 0.46
HSP90AA1 P07900 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
NPC1 O15118 1/20 0.45
RAB9A P51151 1/20 0.45
PARP10 Q53GL7 4/20 0.44
ALDH1A1 P00352 2/20 0.41
PARP4 Q9UKK3 2/20 0.40
PARP1 P09874 2/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
PARP2 Q9UGN5 1/20 0.40
TLR8 Q9NR97 1/20 0.40
HSD17B10 Q99714 2/20 0.40
CYP2C9 P11712 1/20 0.40
TSHR P16473 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6288870 0.85 BDKRB2 (0.44) RAB9AALDH1A1MAPTHSD17B3
SCHEMBL2480571 0.84 RARB (0.50) KMT2AMEN1ALDH1A1TSHRMAPT
SCHEMBL28435445 0.84 KMT2A (0.44) MAPK1KMT2ASMN1; SMN2NPC1RAB9A
SCHEMBL961840 0.83 MAPT (0.47) KMT2AMEN1ALDH1A1CA1CA2
SCHEMBL4766583 0.81 HSD17B3 (0.55) SMN1; SMN2NPC1L3MBTL1HSD17B3
SCHEMBL1983658 0.80 TSHR (0.32) KMT2AMEN1CYP2C9TSHRMAPT
SCHEMBL8979725 0.80 PARP1 (0.46) MAPK1KMT2AMEN1APAF1RGS12
SCHEMBL5952565 0.79 NPC1 (0.50) KMT2AMEN1SMN1; SMN2NPC1RAB9A
SCHEMBL4769427 0.79 PLK1 (0.58) SMN1; SMN2CA1CA2TSHRL3MBTL1
SCHEMBL9596990 0.79 HPGD (0.44) SMN1; SMN2ALDH1A1TLR8EPHX2HSD17B3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5502065-A TREATING HEADACHES PFIZER INC. (US) 1996-03-26 US disclosed
EP-0636129-A1 INDOLE DERIVATIVES AS 5-HT1-LIKE AGONISTS Pfizer Limited (GB) 1995-02-01 EP disclosed
US-5258509-A Catalytic detherification and alkylation BANYU PHARMACEUTICAL CO., LTD. (JP) 1993-11-02 US disclosed
WO-1993021178-A1 INDOLE DERIVATIVES AS 5-HT1-LIKE AGONISTS PFIZER LIMITED (GB) 1993-10-28 WO disclosed
EP-0430037-A2 Process for producing 2-carbon-substituted carbapenem derivatives BANYU PHARMACEUTICAL CO., LTD. (JP) 1991-06-05 EP disclosed