SCHEMBL8980045

SCHEMBL8980045

CC(C)COc1ccnc(CSc2nc3cc(C(F)(F)F)ccc3[nH]2)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 3/20 0.53
NOS3 P29474 2/20 0.53
NOS1 P29475 2/20 0.53
CYP1A2 P05177 10/20 0.42
CYP2D6 P10635 10/20 0.42
CYP2C9 P11712 10/20 0.42
CYP2C19 P33261 10/20 0.42
CYP2E1 P05181 9/20 0.42
CYP3A4 P08684 9/20 0.42
CYP2C8 P10632 9/20 0.42
CYP2B6 P20813 9/20 0.42
RAB9A P51151 3/20 0.40
NPC1 O15118 2/20 0.40
SMN1; SMN2 Q16637 2/20 0.37
POLB P06746 2/20 0.36
MAPT P10636 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
TDP1 Q9NUW8 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980070 0.90 NOS2 (0.55) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL5662514 0.88 NOS2 (0.69) NOS2NOS3NOS1CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL11084434 0.87 NOS2 (0.68) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL8443007 0.84 NOS2 (0.51) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL8980095 0.84 NOS2 (0.51) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL10921896 0.83 NOS2 (0.55) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL2998260 0.83 NOS2 (0.76) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL8980044 0.80 CYP1A2 (0.48) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL6439514 0.78 NOS2 (0.67) NOS2NOS3NOS1CYP1A2CYP2D6
SCHEMBL9526853 0.78 NOS2 (0.67) NOS2NOS3NOS1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0585722-B1 Benzimidazole derivatives as antimicrobal agent against Campylobacter pylon EISAI CO LTD (JP) 1996-05-15 EP disclosed
EP-0585722-A1 Benzimidazole derivatives as antimicrobal agent against Campylobacter pylon Eisai Co., Ltd. (JP) 1994-03-09 EP disclosed