SCHEMBL8980362

SCHEMBL8980362

NC(C(=O)c1ccccc1)C1CCCN1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 8/20 0.48
SLC6A2 P23975 6/20 0.48
SLC6A4 P31645 4/20 0.48
DHFR P00374 1/20 0.45
ALDH1A1 P00352 1/20 0.44
LMNA P02545 1/20 0.44
TSHR P16473 1/20 0.44
TDP1 Q9NUW8 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27682288 0.83 SLC6A3 (0.49) SLC6A3SLC6A2SLC6A4DHFRALDH1A1
SCHEMBL28765067 0.83 SLC6A3 (0.49) SLC6A3SLC6A2SLC6A4DHFRALDH1A1
SCHEMBL8980223 0.78 ALDH1A1 (0.35) SLC6A3SLC6A2SLC6A4DHFRALDH1A1
SCHEMBL27939590 0.77 SLC6A3 (0.44) SLC6A3SLC6A2SLC6A4DHFRALDH1A1
SCHEMBL9081603 0.76 KMT2A (0.48) SLC6A3SLC6A4TSHR
SCHEMBL23383968 0.76 SLC1A2 (0.39) SLC6A3SLC6A2SLC6A4DHFRLMNA
SCHEMBL2267036 0.76 SLC1A2 (0.39) SLC6A3SLC6A2SLC6A4DHFRLMNA
SCHEMBL29291723 0.75 DPP8 (0.51) LMNATDP1
SCHEMBL20833310 0.73 SLC6A2 (0.46) SLC6A3SLC6A2SLC6A4TSHR
SCHEMBL25968626 0.73 SLC6A2 (0.46) SLC6A3SLC6A2SLC6A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103347859-B Synthesis and Anticancer Activity of Aryl and Heteroaryl Quinoline Derivatives EFFICIENT PHARMA MANAGEMENT CORP. (CN) 2015-12-02 CN disclosed
US-5571822-A AMINO-2-PHENYL-4-QUINOLONE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-11-05 US disclosed
WO-1996010563-A1 2-ARYL-4-QUINOLONES AS ANTITUMOR COMPOUNDS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-04-11 WO disclosed