SCHEMBL8980376

SCHEMBL8980376

C=C1C[C@@H]2[C@H](CC[C@]3(C)OCC[C@@H]23)[C@@]2(C)C=CC(=O)C=C12

nearest known ligand 0.65

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 15/20 0.65
KDM4E B2RXH2 1/20 0.65
ALDH1A1 P00352 1/20 0.65
ABCB11 O95342 1/20 0.65
NR3C1 P04150 1/20 0.65
PGR P06401 1/20 0.65
HTR2A P28223 1/20 0.65
OPRK1 P41145 1/20 0.65
HTR2B P41595 1/20 0.65
GUSB P08236 1/20 0.48
LMNA P02545 2/20 0.45
MAPT P10636 2/20 0.45
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980226 0.88 GUSB (0.62) CYP19A1KDM4EALDH1A1ABCB11NR3C1
SCHEMBL11980206 0.80 CYP19A1 (0.84) CYP19A1KDM4EALDH1A1ABCB11NR3C1
SCHEMBL13817790 0.80 CYP19A1 (0.69) CYP19A1KDM4EALDH1A1ABCB11NR3C1
SCHEMBL9255515 0.80 CYP19A1 (0.69) CYP19A1KDM4EALDH1A1ABCB11NR3C1
SCHEMBL8980330 0.79 CYP19A1 (0.68) CYP19A1KDM4EALDH1A1ABCB11NR3C1
SCHEMBL8980318 0.79 CYP19A1 (0.71) CYP19A1KDM4EALDH1A1ABCB11NR3C1
Exemestane SCHEMBL6215 0.79 CYP19A1 (1.00) CYP19A1KDM4EALDH1A1ABCB11NR3C1
Exemestane SCHEMBL19452231 0.79 CYP19A1 (1.00) CYP19A1KDM4EALDH1A1ABCB11NR3C1
Exemestane SCHEMBL13794245 0.79 CYP19A1 (1.00) CYP19A1KDM4EALDH1A1ABCB11NR3C1
Exemestane SCHEMBL172860 0.79 CYP19A1 (1.00) CYP19A1KDM4EALDH1A1ABCB11NR3C1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519051-A AROMATASE INHIBITORS USEFUL FOR TREATMENT OF DISEASES CAUSED BY EXCESS OF ESTROGEN, FOR EXAMPLE, BREAST CANCER, UTERINE CANCER TEIKOKU HORMONE MFG. CO., LTD. (JP) 1996-05-21 US disclosed
EP-0582713-A1 NOVEL OXA- OR AZASTEROID DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1994-02-16 EP disclosed