SCHEMBL8980226

SCHEMBL8980226

C[C@]12C=CC(=O)C=C1C(=O)C[C@@H]1[C@@H]2CC[C@]2(C)OCC[C@@H]12

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
GUSB P08236 1/20 0.62
CYP19A1 P11511 15/20 0.49
KDM4E B2RXH2 1/20 0.49
ALDH1A1 P00352 1/20 0.49
ABCB11 O95342 1/20 0.49
NR3C1 P04150 1/20 0.49
PGR P06401 1/20 0.49
HTR2A P28223 1/20 0.49
OPRK1 P41145 1/20 0.49
HTR2B P41595 1/20 0.49
LMNA P02545 2/20 0.46
MAPT P10636 2/20 0.46
CYP3A4 P08684 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8980376 0.88 CYP19A1 (0.65) GUSBCYP19A1KDM4EALDH1A1ABCB11
SCHEMBL8980363 0.79 CYP19A1 (0.72) CYP19A1LMNAMAPTCYP3A4
SCHEMBL8980211 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1NR3C1PGRLMNA
SCHEMBL8980219 0.77 CYP19A1 (0.67) CYP19A1ALDH1A1NR3C1PGRLMNA
SCHEMBL13518386 0.75 GUSB (0.75) GUSBCYP19A1KDM4EALDH1A1ABCB11
SCHEMBL11112810 0.75 GUSB (0.61) GUSBCYP19A1KDM4EALDH1A1ABCB11
SCHEMBL11425309 0.74 GUSB (0.60) GUSBCYP19A1KDM4EALDH1A1ABCB11
SCHEMBL6524579 0.74 GUSB (0.60) GUSBCYP19A1KDM4EALDH1A1ABCB11
SCHEMBL11137065 0.74 GUSB (0.60) GUSBCYP19A1KDM4EALDH1A1ABCB11
SCHEMBL9240286 0.74 GUSB (0.60) GUSBCYP19A1KDM4EALDH1A1ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5519051-A AROMATASE INHIBITORS USEFUL FOR TREATMENT OF DISEASES CAUSED BY EXCESS OF ESTROGEN, FOR EXAMPLE, BREAST CANCER, UTERINE CANCER TEIKOKU HORMONE MFG. CO., LTD. (JP) 1996-05-21 US disclosed
EP-0582713-A1 NOVEL OXA- OR AZASTEROID DERIVATIVE TEIKOKU HORMONE MFG. CO., LTD. (JP) 1994-02-16 EP disclosed