SCHEMBL8980467

SCHEMBL8980467

CC(=O)NCC(=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.62

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.62
CES2 O00748 1/20 0.57
CES1 P23141 1/20 0.57
TP53 P04637 1/20 0.55
KMT2A Q03164 3/20 0.54
TSHR P16473 2/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
KMO O15229 1/20 0.53
HPGD P15428 2/20 0.53
LMNA P02545 1/20 0.53
L3MBTL1 Q9Y468 1/20 0.53
MEN1 O00255 2/20 0.52
AGTR1 P30556 1/20 0.52
POLB P06746 1/20 0.51
MAPT P10636 1/20 0.51
BLM P54132 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17790237 0.85 ALDH1A1 (0.61) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL38656427 0.83 ALDH1A1 (0.68) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL27570821 0.83 ALDH1A1 (0.68) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL8921654 0.83 ALDH1A1 (0.68) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL11153162 0.83 ALDH1A1 (0.57) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL10806282 0.82 ATM (0.55) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL4472065 0.81 SMN1; SMN2 (0.58) ALDH1A1CES1KMT2ATSHRSMN1; SMN2
SCHEMBL23014104 0.81 ALDH1A1 (0.77) ALDH1A1TP53KMT2ASMN1; SMN2HPGD
SCHEMBL17788611 0.81 ADRB2 (0.58) ALDH1A1CES2CES1TP53KMT2A
SCHEMBL8298069 0.81 ALDH1A1 (0.70) ALDH1A1CES2CES1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5571822-A AMINO-2-PHENYL-4-QUINOLONE DERIVATIVES THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-11-05 US disclosed
WO-1996010563-A1 2-ARYL-4-QUINOLONES AS ANTITUMOR COMPOUNDS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1996-04-11 WO disclosed
EP-0094727-A2 Substituted heterocyclyl phenylformamidines, processes for their preparation and their pharmaceutical use ISTITUTO DE ANGELI S.p.A. (IT) 1983-11-23 EP disclosed