SCHEMBL8980924

SCHEMBL8980924

CCCCON(C[Si](C)(C)C)C(C)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 2/20 0.36
POLB P06746 2/20 0.35
SIGMAR1 Q99720 1/20 0.34
GPR88 Q9GZN0 2/20 0.34
CALM1 P0DP23 1/20 0.34
CDC7 O00311 1/20 0.33
PLK4 O00444 1/20 0.33
CHEK1 O14757 1/20 0.33
CHUK O15111 1/20 0.33
PDPK1 O15530 1/20 0.33
DYRK3 O43781 1/20 0.33
ROCK2 O75116 1/20 0.33
PRKD3 O94806 1/20 0.33
MAP4K4 O95819 1/20 0.33
PAK4 O96013 1/20 0.33
NTRK1 P04629 1/20 0.33
PRKCG P05129 1/20 0.33
INSR P06213 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6958572 0.77 LTA4H (0.37) LTA4HPOLBGPR88ALDH1A1
SCHEMBL4716852 0.77 LTA4H (0.37) LTA4HPOLBGPR88ALDH1A1
SCHEMBL9265557 0.71 LTA4H (0.36) LTA4HPOLBSIGMAR1GPR88CALM1
SCHEMBL2206565 0.66 ADRA2A (0.36) ALDH1A1ADRA2AADRA2BADRA2CHTR2A
SCHEMBL1773270 0.66 ADRA2A (0.36) ALDH1A1ADRA2AADRA2BADRA2CHTR2A
SCHEMBL1773267 0.66 ADRA2A (0.36) ALDH1A1ADRA2AADRA2BADRA2CHTR2A
Isopropylbenzene SCHEMBL28865209 0.65 LTA4H (0.46) LTA4HPOLBGPR88MAPK1ALDH1A1
SCHEMBL28859344 0.65 TSHR (0.46) LTA4HPOLBGPR88ALDH1A1
SCHEMBL159324 0.65 LTA4H (0.46) LTA4HPOLBGPR88ALDH1A1ADRA2A
SCHEMBL14314047 0.65 LTA4H (0.46) LTA4HPOLBGPR88ALDH1A1ADRA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711280-A1 PERHYDROISOINDOLE DERIVATIVES AS P SUBSTANCE ANTAGONISTS Aventis Pharma S.A. (FR) 1996-05-15 EP disclosed
US-5451601-A Perhydroisoindole derivatives and pharmaceutical compositions containing them RHONE-POULENC RORER S.A. (FR) 1995-09-19 US disclosed
WO-1995004040-A1 PERHYDROISOINDOLE DERIVATIVES AS P SUBSTANCE ANTAGONISTS RHONE-POULENC RORER S.A. (FR) 1995-02-09 WO disclosed