SCHEMBL8981985

SCHEMBL8981985

NC(=O)CN1CCCCc2ccccc21

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 4/20 0.67
CHRM4 P08173 4/20 0.67
CHRM1 P11229 4/20 0.67
CHRM3 P20309 4/20 0.67
ALDH1A1 P00352 8/20 0.65
GAA P10253 3/20 0.65
MAPT P10636 5/20 0.59
KDM4E B2RXH2 3/20 0.59
MEN1 O00255 3/20 0.59
KMT2A Q03164 3/20 0.59
HPGD P15428 1/20 0.59
ALOX15 P16050 1/20 0.59
TSHR P16473 1/20 0.59
CASP1 P29466 1/20 0.59
CASP7 P55210 1/20 0.59
TDP1 Q9NUW8 1/20 0.59
HDAC1 Q13547 2/20 0.54
HDAC6 Q9UBN7 2/20 0.54
HDAC8 Q9BY41 1/20 0.54
ALPL P05186 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4700798 0.95 ALDH1A1 (0.71) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL6025353 0.89 ALDH1A1 (0.62) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL2991784 0.86 CHRM2 (0.68) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL30775585 0.86 CHRM2 (0.68) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL1102038 0.81 CHRM2 (0.70) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL29930459 0.80 CHRM2 (1.00) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL28643439 0.80 CHRM2 (1.00) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL11881953 0.79 ALDH1A1 (0.62) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL9974151 0.79 CHRM2 (0.68) CHRM2CHRM4CHRM1CHRM3ALDH1A1
SCHEMBL29930254 0.79 CHRM2 (1.00) CHRM2CHRM4CHRM1CHRM3ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0711283-A1 TETRAHYDRO-1H-BENZAZEPINONES AND HEXAHYDROAZEPINONES AS SELECTIVE CHOLECYSTOKININ-B RECEPTOR ANTAGONISTS PFIZER INC. (US) 1996-05-15 EP disclosed
WO-1995003281-A1 TETRAHYDRO-1H-BENZAZEPINONES AND HEXAHYDROAZEPINONES AS SELECTIVE CHOLECYSTOKININ-B RECEPTOR ANTAGONISTS PFIZER INC. (US) 1995-02-02 WO disclosed
EP-0322779-A2 Benzolactam compounds and pharmaceutical uses thereof Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-07-05 EP disclosed