SCHEMBL8982437

SCHEMBL8982437

COC(=O)c1ccc(CCCC(C(C#N)C#N)C(OC)OC)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP4A11 Q02928 2/20 0.54
CYP4F2 P78329 1/20 0.52
LOXL2 Q9Y4K0 1/20 0.43
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2C9 P11712 1/20 0.40
HPGD P15428 1/20 0.40
ALOX15 P16050 1/20 0.40
ALOX12 P18054 1/20 0.40
CYP2C19 P33261 1/20 0.40
CKS1B P61024 1/20 0.40
SKP2 Q13309 1/20 0.40
HIF1A Q16665 1/20 0.40
HSD17B10 Q99714 1/20 0.40
IDH1 O75874 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9088289 0.89 CYP4A11 (0.41) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL9087966 0.89 CA12 (0.41) CYP4A11CYP4F2ALDH1A1CYP1A2CYP3A4
SCHEMBL9086571 0.85 CYP4A11 (0.42) CYP4A11CYP4F2ALDH1A1HRH1MAPT
SCHEMBL27319129 0.83 ALDH1A1 (0.41) CYP4A11CYP4F2ALDH1A1HSD17B10HRH1
SCHEMBL9085713 0.81 CA12 (0.39) CYP4A11CYP4F2CA1CA2CA12
SCHEMBL27323755 0.79 ALDH1A1 (0.43) CYP4A11CYP4F2LOXL2ALDH1A1TP53
SCHEMBL9050346 0.79 CYP4A11 (0.61) CYP4A11CYP4F2LOXL2ALDH1A1TP53
SCHEMBL20504197 0.78 CYP4A11 (0.66) CYP4A11CYP4F2LOXL2ALDH1A1TP53
SCHEMBL9206449 0.78 CYP4A11 (0.66) CYP4A11CYP4F2LOXL2ALDH1A1TP53
SCHEMBL10169575 0.76 CYP4A11 (0.68) CYP4A11CYP4F2LOXL2ALDH1A1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5496822-A Compounds and methods for treating tumors TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-03-05 US disclosed
EP-0434426-A1 Condensed heterocyclic compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1991-06-26 EP disclosed