Phenamet

Phenamet

SCHEMBL8986

CCOC(=O)C(CCSC)NC(=O)Cc1ccc(N(CCCl)CCCl)cc1

nearest known ligand 0.53

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.53
PPID Q08752 1/20 0.49
LMNA P02545 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.43
POLB P06746 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
CNR2 P34972 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
DRD1 P21728 1/20 0.39
HTT P42858 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MEN1 O00255 1/20 0.39
USP2 O75604 1/20 0.39
TAS1R3 Q7RTX0 1/20 0.39
TAS1R1 Q7RTX1 1/20 0.39
ABCB11 O95342 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CHRM2 P08172 1/20 0.38
CYP3A4 P08684 1/20 0.38
ADRA2A P08913 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Phenamet SCHEMBL8985 1.00 KMT2A (0.53) KMT2APPIDLMNAL3MBTL1POLB
Phenamet SCHEMBL23493623 0.91 KMT2A (0.45) KMT2APPIDLMNAL3MBTL1POLB
SCHEMBL2330760 0.81 PPID (0.55) PPIDL3MBTL1POLBCNR2
SCHEMBL2330757 0.81 PPID (0.55) PPIDL3MBTL1POLBCNR2
SCHEMBL8726309 0.79 KMT2A (0.61) KMT2ALMNAL3MBTL1POLBNPSR1
SCHEMBL11127008 0.77 SMN1; SMN2 (0.46) KMT2APPIDLMNASMN1; SMN2DRD1
Hydrochloric Acid SCHEMBL11124542 0.77 SMN1; SMN2 (0.45) KMT2APPIDLMNASMN1; SMN2DRD1
SCHEMBL11124423 0.75 LMNA (0.42) PPIDLMNASMN1; SMN2
SCHEMBL7906473 0.74 KMT2A (0.52) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL8744707 0.73 LMNA (0.51) PPIDLMNAL3MBTL1POLBNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 21211 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4748859-A2 CHEMICALLY AND PHOTOCHEMICALLY INITIATED CELL MEMBRANE BLEBBING TO INDUCE CELL VESICLE PRODUCTION, MODIFICATIONS THEREOF, AND USES THEREOF The Regents of the University of California (US) 2026-05-27 EP claimed
US-20260137794-A1 LIGAND-DRUG CONJUGATE AND USE THEREOF SYSTIMMUNE INC (US) 2026-05-21 US claimed
EP-4743490-A1 HUMANIZED ANTI-CD7 ANTIBODY Christian-Albrechts-Universität zu Kiel (DE) 2026-05-20 EP claimed
WO-2026099502-A1 NOVEL DRUG CONJUGATES FOR TESTING CELLULAR DRUG UPTAKE Deutsches Krebsforschungszentrum Stiftung des öffentlichen Rechts (DE) 2026-05-15 WO claimed
US-20260108619-A1 CONJUGATION LINKERS, CELL BINDING MOLECULE-DRUG CONJUGATES CONTAINING THE LINKERS, METHODS OF MAKING AND USES SUCH CONJUGATES WITH THE LINKERS HANGZHOU DAC BIOTECH CO., LTD. (CN) 2026-04-23 US claimed
US-20260085100-A1 METHODS OF ANTIGEN PRODUCTION THE WISTAR INSTITUTE OF ANATOMY AND BIOLOGY (US) 2026-03-26 US claimed
US-12576124-B2 Formulation of a conjugate of a tubulysin analog to a cell-binding molecule HANGZHOU DAC BIOTECH CO., LTD (CN) 2026-03-17 US claimed
EP-4698185-A1 METHODS AND SYSTEMS FOR IMPROVING ANTI-CANCER THERAPIES Osasuna Therapeutics SA (CH) 2026-02-25 EP claimed
EP-4694909-A1 METHODS OF MODULATING THE EPITHELIAL-MESENCHYMAL TRANSITION RS Oncology, LLC (US) 2026-02-18 EP claimed
EP-4687999-A1 TROP2 CONJUGATED BIOLOGICAL MOLECULES, PHARMACEUTICAL COMPOSITIONS AND METHODS OBI Pharma, Inc. (TW) 2026-02-11 EP claimed
US-20020009444-A1 Intrathecal administration of rituximab for treatment of central nervous system lymphomas IDEC PHARMACEUTICALS CORPORATION (US) 2002-01-24 US claimed
WO-2001080884-A1 INTRATHECAL ADMINISTRATION OF RITUXIMAB FOR TREATMENT OF CENTRAL NERVOUS SYSTEM LYMPHOMAS IDEC PHARMACEUTICALS CORPORATION (US) 2001-11-01 WO claimed
CN-1294519-A Pharmaceutical composition containing a compound having an activity of promoting the absorption of an active ingredient INPHARMA SA (CH) 2001-05-09 CN claimed
EP-1083896-A1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 2001-03-21 EP claimed
EP-1073470-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2001-02-07 EP claimed
WO-2000054795-A1 COMBINED THERAPY WITH A CHEMOTHERAPEUTIC AGENT AND AN ONCOLYTIC VIRUS FOR KILLING TUMOR CELLS IN A SUBJECT THE TRUSTEES OF THE UNIVERSITY OF PENNSYLVANIA (US) 2000-09-21 WO claimed
WO-2000048636-A1 PHARMACEUTICAL COMPOSITIONS CONTAINING COMPOUNDS WITH ACTIVITY FOR THE ENHANCEMENT OF ABSORPTION OF ACTIVE INGREDIENTS INPHARMA S.A. (CH) 2000-08-24 WO claimed
WO-2000040269-A2 PHARMACEUTICAL COMPOSITIONS FOR TREATMENT OF DISEASED TISSUES LEE CLARENCE C (US) 2000-07-13 WO claimed
WO-1999058126-B1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES ENDOWMENT RES INHUMAN BIOLOGY (US) 2000-02-17 WO claimed
WO-1999058126-A1 USE OF NEOMYCIN FOR TREATING ANGIOGENESIS-RELATED DISEASES THE ENDOWMENT FOR RESEARCH IN HUMAN BIOLOGY, INC. (US) 1999-11-18 WO claimed