SCHEMBL8726309

SCHEMBL8726309

CCOC(=O)CCC(NC(=O)Cc1ccc(N(CCCl)CCCl)cc1)C(=O)O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.61
LMNA P02545 3/20 0.52
L3MBTL1 Q9Y468 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
CNR2 P34972 3/20 0.43
CYP3A4 P08684 3/20 0.43
ALDH1A1 P00352 3/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
HIF1A Q16665 3/20 0.43
ALOX15 P16050 2/20 0.43
NFKB1 P19838 2/20 0.43
THPO P40225 2/20 0.43
MAPT P10636 2/20 0.43
PMP22 Q01453 2/20 0.43
MEN1 O00255 2/20 0.43
ABCB11 O95342 1/20 0.43
CHRM2 P08172 1/20 0.43
ADRA2A P08913 1/20 0.43
CHRM1 P11229 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8723902 0.90 KMT2A (0.64) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL8723896 0.86 KMT2A (0.69) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL7900436 0.86 KMT2A (0.69) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL8727524 0.84 KMT2A (0.67) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL7906473 0.80 KMT2A (0.52) KMT2ALMNAL3MBTL1NPSR1CNR2
Phenamet SCHEMBL8985 0.79 KMT2A (0.53) KMT2ALMNAL3MBTL1NPSR1CNR2
Phenamet SCHEMBL8986 0.79 KMT2A (0.53) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL14497664 0.79 NPSR1 (0.59) KMT2ALMNAL3MBTL1NPSR1CNR2
Alalon SCHEMBL31687764 0.76 KMT2A (0.65) KMT2ALMNAL3MBTL1NPSR1CNR2
SCHEMBL7719488 0.74 KMT2A (0.49) KMT2ALMNACYP3A4ALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0651740-B1 AMINO ACID LINKED NITROGEN MUSTARD DERIVATIVES AND THEIR USE AS PRODRUGS IN THE TREATMENT OF TUMOURS ZENECA LTD (GB) 1998-10-21 EP claimed
EP-0651740-B1 AMINO ACID LINKED NITROGEN MUSTARD DERIVATIVES AND THEIR USE AS PRODRUGS IN THE TREATMENT OF TUMOURS ZENECA LTD (GB) 1998-10-21 EP disclosed