SCHEMBL898618

SCHEMBL898618

CC(C)N=C=NC(C)C.CCCN=C=NCCC

nearest known ligand 0.32

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25895367 0.92
SCHEMBL132315 0.81
SCHEMBL9074979 0.79 CYP1A2 (0.38) TRPA1TRPV1CYP1A2CYP2D6
SCHEMBL1005697 0.78 NAAA (0.38) TRPA1TRPV1CYP1A2CYP2D6
SCHEMBL3626821 0.75 CYP1A2 (0.32) CYP1A2CYP2D6
SCHEMBL9064503 0.75 NAAA (0.50) CYP1A2CYP2D6
SCHEMBL27916922 0.74 TRPA1 (0.50) TRPA1TRPV1
SCHEMBL6720 0.74
Dimethylamine SCHEMBL8019309 0.73 CYP1A2 (0.34) TRPA1TRPV1CYP1A2CYP2D6
SCHEMBL26926038 0.73

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012042534-A2 PROCESSES FOR THE PREPARATION OF R-SITAGLIPTIN AND INTERMEDIATES THEREOF GLENMARK GENERICS LIMITED (IN) 2012-04-05 WO claimed
WO-2012042534-A2 PROCESSES FOR THE PREPARATION OF R-SITAGLIPTIN AND INTERMEDIATES THEREOF GLENMARK GENERICS LIMITED (IN) 2012-04-05 WO disclosed