SCHEMBL8987641

SCHEMBL8987641

CN(CCCC#N)Cc1ccc(Cl)cc1

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PYCR1 P32322 2/20 0.51
TMEM97 Q5BJF2 5/20 0.51
SIGMAR1 Q99720 5/20 0.51
KDM4E B2RXH2 1/20 0.46
TSHR P16473 1/20 0.46
POLB P06746 1/20 0.43
DPP7 Q9UHL4 1/20 0.41
P2RX7 Q99572 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL149999 0.83 SIGMAR1 (0.59) PYCR1TMEM97SIGMAR1TSHR
SCHEMBL8987611 0.83 NPC1 (0.42) PYCR1DPP7
SCHEMBL9131306 0.79 TMEM97 (0.56) PYCR1TMEM97SIGMAR1KDM4ETSHR
SCHEMBL11932509 0.78 SIGMAR1 (0.52) PYCR1TMEM97SIGMAR1KDM4ETSHR
SCHEMBL31612490 0.77 SIGMAR1 (0.55) PYCR1TMEM97SIGMAR1KDM4ETSHR
SCHEMBL9266697 0.76 LSS (0.44) TMEM97SIGMAR1
SCHEMBL17917694 0.76 SIGMAR1 (0.54) PYCR1TMEM97SIGMAR1KDM4ETSHR
SCHEMBL7855920 0.75 SIGMAR1 (0.50) PYCR1TMEM97SIGMAR1KDM4ETSHR
SCHEMBL18532755 0.75 PYCR1 (0.67) PYCR1TMEM97SIGMAR1KDM4ETSHR
SCHEMBL8987565 0.75 KCNH2 (0.46)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5527955-A AGONIST OF GAMMA AMINOBUTYRIC ACID JOHN WYETH & BROTHER, LIMITED (GB) 1996-06-18 US disclosed
EP-0345068-B1 Agonist of gamma-aminobutyric acid WYETH JOHN & BROTHER LTD (GB) 1995-03-15 EP disclosed
US-5321047-A Antidepressant JOHN WYETH & BROTHER, LIMITED (GB) 1994-06-14 US disclosed
EP-0345068-A2 Agonist of gamma-aminobutyric acid JOHN WYETH & BROTHER LIMITED (GB) 1989-12-06 EP disclosed