SCHEMBL8988145

SCHEMBL8988145

CC(=O)Oc1cc2c(c(O)c1O)[C@H]1CC[C@]3(C)CCC[C@H]3[C@@H]1[C@H](C)C2

nearest known ligand 0.36

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
SHBG P04278 1/20 0.36
STS P08842 2/20 0.33
PTPN1 P18031 1/20 0.32
MEN1 O00255 1/20 0.30
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8988016 0.83 CYP19A1 (0.40) SHBGSTSMAPT
SCHEMBL8987956 0.73 SHBG (0.38) SHBGSTSPTPN1MEN1MAPT
SCHEMBL4816847 0.71 ESR1 (0.37) SHBGSTSMEN1MAPTMAPK1
SCHEMBL8518605 0.70 ESR1 (0.38) SHBGPTPN1
SCHEMBL11981697 0.70 SHBG (0.62) SHBGSTSMEN1MAPTKMT2A
SCHEMBL17296147 0.69 ESR1 (0.37) SHBGPTPN1
SCHEMBL5851260 0.69 SHBG (0.61) SHBGSTSMEN1MAPTMAPK1
SCHEMBL6130909 0.67 STS (0.48) SHBGSTSKMT2A
SCHEMBL8969620 0.67 CYP19A1 (0.54) SHBGSTSMAPT
SCHEMBL4588126 0.66 SHBG (0.56) SHBGSTSMEN1MAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0719276-A1 ORALLY ACTIVE DERIVATIVES OF 1,3,5(10)-ESTRATRIENE THE GOVERNMENT OF THE UNITED STATES OF AMERICA as represented by the SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES (US) 1996-07-03 EP disclosed